SCHEMBL9501155

SCHEMBL9501155

CN1CCN(c2cc3c(c(N)c2F)c(=O)c(C(=O)O)cn3C2CC2)CC1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 2/20 0.57
HRH3 Q9Y5N1 1/20 0.57
ALDH1A1 P00352 4/20 0.54
KDM4E B2RXH2 3/20 0.54
LMNA P02545 3/20 0.53
HPGD P15428 2/20 0.53
HSD17B10 Q99714 2/20 0.53
CACNA1F O60840 1/20 0.53
POLB P06746 1/20 0.53
MAPK1 P28482 1/20 0.53
CACNA1D Q01668 1/20 0.53
CACNA1S Q13698 1/20 0.53
CACNA1C Q13936 1/20 0.53
MAPT P10636 1/20 0.53
GSK3B P49841 4/20 0.52
TOP2A P11388 2/20 0.51
TOP2B Q02880 2/20 0.51
CYP1A2 P05177 1/20 0.51
CYP2C9 P11712 1/20 0.51
MEN1 O00255 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9501344 0.91 KCNH2 (0.62) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL8556904 0.89 KCNH2 (0.71) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL9023279 0.88 KDM4E (0.67) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL9501991 0.85 KCNH2 (0.71) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL9023644 0.85 KCNH2 (0.58) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL9500959 0.85 KCNH2 (0.71) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL9023635 0.85 KCNH2 (0.58) KCNH2HRH3ALDH1A1KDM4ELMNA
SCHEMBL10685966 0.85 KCNH2 (0.58) KCNH2HRH3ALDH1A1KDM4ELMNA
Hydrochloric Acid SCHEMBL9504778 0.84 KCNH2 (0.69) KCNH2HRH3ALDH1A1KDM4ELMNA
Hydrochloric Acid SCHEMBL9504788 0.84 KCNH2 (0.69) KCNH2HRH3ALDH1A1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0312085-B1 NOVEL QUINOLINE DERIVATIVES, PROCESSES FOR PREPARATION THEREOF AND ANTIBACTERIAL AGENT CONTAINING THEM Dainippon Pharmaceutical Co., Ltd. (JP) 1993-05-12 EP disclosed
US-5164392-A Active against streptococci and staphylococci DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1992-11-17 US disclosed
US-5013841-A Oxo quinoline derivatives DAINIPPON PHARMACEUTICAL CO., LTD. (JP) 1991-05-07 US disclosed
EP-0312085-A2 Novel quinoline derivatives, processes for preparation thereof and antibacterial agent containing them Dainippon Pharmaceutical Co., Ltd. (JP) 1989-04-19 EP disclosed