SCHEMBL9501335

SCHEMBL9501335

CC1CN(Cc2ccncc2)c2ccccc21

nearest known ligand 0.54

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CACNA1I Q9P0X4 11/20 0.54
ALOX12 P18054 1/20 0.47
CACNA1G O43497 12/20 0.45
CACNA1H O95180 11/20 0.45
GRM2 Q14416 1/20 0.44
NOTUM Q6P988 1/20 0.42
BRD4 O60885 1/20 0.42
ROCK1 Q13464 1/20 0.42
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13227810 0.75 NOTUM (0.50) CACNA1IALOX12CACNA1GCACNA1HNOTUM
SCHEMBL3553533 0.74 ALOX15 (0.43) CACNA1IALOX12CACNA1GCACNA1HNOTUM
SCHEMBL8202698 0.74 TAAR1 (0.54)
SCHEMBL3553536 0.74 ALOX15 (0.43) CACNA1IALOX12CACNA1GCACNA1HNOTUM
SCHEMBL5870956 0.74 SIRT2 (0.47) CACNA1ICACNA1GCACNA1HGRM2
SCHEMBL20879389 0.74 HDAC6 (0.55)
SCHEMBL7695554 0.74 SIRT2 (0.51) ALOX12NOTUMBRD4
SCHEMBL17846769 0.74 CACNA1I (0.44) CACNA1ICACNA1GCACNA1H
SCHEMBL6684665 0.73 PRCP (0.45) ALOX12NOTUMROCK1DRD2DRD4
SCHEMBL26091678 0.72 CACNA1I (0.41) CACNA1ICACNA1GCACNA1HBRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5214058-A Acetylcholinesterase inhibitors, treatment of senile dementia HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1993-05-25 US disclosed
EP-0471296-A1 1-(Pyridinylalkyl)-1H-indoles, indolines and related analogs HOECHST-ROUSSEL PHARMACEUTICALS INCORPORATED (US) 1992-02-19 EP disclosed