SCHEMBL9501944

SCHEMBL9501944

CCCC(=O)Oc1c(-c2ccc(-c3ccccc3)cc2)nc2ccccc2c1C(=O)O

nearest known ligand 0.59

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 9/20 0.59
PDE10A Q9Y233 4/20 0.54
TSHR P16473 1/20 0.54
LMNA P02545 2/20 0.52
CYP2D6 P10635 1/20 0.51
CYP2C19 P33261 1/20 0.51
POLB P06746 1/20 0.50
TACR3 P29371 4/20 0.48
TACR2 P21452 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9502807 0.85 DHODH (0.64) DHODHPDE10ATSHRLMNACYP2D6
SCHEMBL5498214 0.82 PDE10A (0.62) DHODHPDE10ATSHRLMNACYP2D6
SCHEMBL9505258 0.82 DHODH (0.69) DHODHPDE10A
SCHEMBL10559127 0.81 DHODH (0.67) DHODHPDE10A
SCHEMBL3959255 0.79 TACR3 (0.68) DHODHPDE10ATSHRLMNACYP2D6
SCHEMBL14492079 0.74 PDE10A (0.68) DHODHPDE10ATSHRLMNACYP2D6
SCHEMBL4234246 0.74 DHODH (0.57) DHODHPDE10ATSHRLMNACYP2D6
SCHEMBL4897475 0.73 TACR3 (0.68) DHODHPDE10ATSHRLMNACYP2D6
SCHEMBL5496908 0.73 SMN1; SMN2 (0.56) DHODHPDE10ATSHRLMNATACR3
SCHEMBL9501979 0.73 DHODH (1.00) DHODHPDE10ATSHRLMNACYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0305952-B1 SUBSTITUTED 2-PHENYL-4-QUINOLINE-CARBOXYLIC ACIDS AMERICAN CYANAMID COMPANY (US) 1993-06-02 EP disclosed
US-4847381-A ANTIARTHRITIC AGENTS AMERICAN CYANAMID COMPANY (US) 1989-07-11 US disclosed
EP-0305952-A1 Substituted 2-phenyl-4-quinoline-carboxylic acids AMERICAN CYANAMID COMPANY (US) 1989-03-08 EP disclosed