SCHEMBL9502193

SCHEMBL9502193

COC(=O)c1ccc(-c2ncc[nH]2)c(N)c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 11/20 0.65
ALDH1A1 P00352 8/20 0.65
HPGD P15428 6/20 0.51
MAPT P10636 5/20 0.51
GAA P10253 2/20 0.51
HSD17B10 Q99714 2/20 0.51
GLA P06280 1/20 0.51
CASP1 P29466 1/20 0.51
CASP7 P55210 1/20 0.51
ATM Q13315 1/20 0.51
NPSR1 Q6W5P4 2/20 0.46
NPC1 O15118 2/20 0.46
RAB9A P51151 2/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
USP2 O75604 1/20 0.45
CSNK1A1 P48729 1/20 0.43
TYRO3 Q06418 1/20 0.43
DYRK1B Q9Y463 1/20 0.43
ALOX15 P16050 3/20 0.43
HTT P42858 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31238771 1.00 KDM4E (0.65) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL1485475 0.86 KDM4E (0.68) KDM4EALDH1A1HPGDMAPTGAA
SCHEMBL1485283 0.84 KDM4E (0.67) KDM4EALDH1A1HPGDMAPTHSD17B10
SCHEMBL31521365 0.83 KDM4E (0.65) KDM4EALDH1A1NPC1RAB9ACSNK1A1
SCHEMBL16862868 0.83 KDM4E (0.65) KDM4EALDH1A1GAACSNK1A1TYRO3
SCHEMBL16862898 0.83 KDM4E (0.65) KDM4EALDH1A1CSNK1A1TYRO3DYRK1B
SCHEMBL22530491 0.82 KDM4E (0.63) KDM4EALDH1A1CSNK1A1TYRO3DYRK1B
SCHEMBL29140743 0.79 KDM4E (1.00) KDM4EALDH1A1HPGDMAPTNPC1
SCHEMBL9503741 0.79 ALDH1A1 (0.59) KDM4EALDH1A1HPGDMAPTNPSR1
SCHEMBL3062520 0.78 KDM4E (0.70) KDM4EALDH1A1KDM6BKDM5CKDM4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-117980307-A Substituted tricyclic compounds as PARP inhibitors and application thereof 上海瑛派药业有限公司 2024-05-03 CN disclosed
EP-0543865-A1 BENZAMIDE DERIVATIVES RHONE-POULENC RORER LIMITED (GB) 1993-06-02 EP disclosed