SCHEMBL9502346

SCHEMBL9502346

C=CCOC(=O)C1=C(C)NC(CSCc2ccccc2)=C(C(=O)OC(C)(C)C)C1c1cccc(Cl)c1Cl

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 4/20 0.47
MEN1 O00255 4/20 0.47
KMT2A Q03164 4/20 0.47
KDM4E B2RXH2 4/20 0.47
MAPT P10636 4/20 0.47
CYP3A4 P08684 3/20 0.47
CYP2C19 P33261 3/20 0.47
HSD17B10 Q99714 3/20 0.47
ABCB11 O95342 3/20 0.47
LMNA P02545 3/20 0.47
ADORA3 P0DMS8 3/20 0.47
OPRK1 P41145 3/20 0.47
ALDH1A1 P00352 3/20 0.47
TBXA2R P21731 3/20 0.47
ADRA1A P35348 3/20 0.47
SLC6A3 Q01959 3/20 0.47
CYP1A2 P05177 2/20 0.47
HIF1A Q16665 2/20 0.47
NR1I2 O75469 2/20 0.47
PGR P06401 2/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9504224 0.86 KDM4E (0.61) CYP2C9MEN1KMT2AKDM4EMAPT
SCHEMBL9502226 0.81 KDM4E (0.47) CYP2C9MEN1KMT2AKDM4EMAPT
SCHEMBL7473385 0.78 TBXA2R (0.60) CYP2C9MEN1KMT2AKDM4EMAPT
SCHEMBL3027068 0.76 CYP2C9 (0.65) CYP2C9MEN1KMT2AKDM4EMAPT
SCHEMBL9501245 0.75 CYP2C9 (0.62) CYP2C9MEN1KMT2AKDM4EMAPT
SCHEMBL8510425 0.74 CYP2C9 (0.60) CYP2C9MEN1KMT2AKDM4EMAPT
SCHEMBL7428857 0.74 CYP2C9 (0.64) CYP2C9MEN1KMT2AKDM4EMAPT
SCHEMBL3023501 0.74 KDM4E (0.60) CYP2C9MEN1KMT2AKDM4EMAPT
SCHEMBL9505249 0.73 ALDH1A1 (0.67) MEN1KMT2AKDM4EMAPTHSD17B10
SCHEMBL10747093 0.72 CYP2C9 (0.73) CYP2C9MEN1KMT2AKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458823-B1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-10-13 EP disclosed
US-5245039-A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA (IT) 1993-09-14 US disclosed
WO-1990009376-A1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-23 WO disclosed
EP-0383320-A1 A process for preparation of enantiomerically pure polysubstituted 1,4-dihydropyridines BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1990-08-22 EP disclosed