SCHEMBL9505249

SCHEMBL9505249

C=CCOC(=O)C1=C(C)NC(C)=C(C(=O)OC(C)(C)C)C1c1ccccc1

nearest known ligand 0.67

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.67
KDM4E B2RXH2 3/20 0.67
HSD17B10 Q99714 2/20 0.67
HPGD P15428 2/20 0.67
TP53 P04637 2/20 0.67
MAPT P10636 3/20 0.60
MEN1 O00255 2/20 0.60
KMT2A Q03164 2/20 0.60
LMNA P02545 1/20 0.60
GAA P10253 1/20 0.60
MAPK1 P28482 1/20 0.60
CACNA1B Q00975 7/20 0.58
CA1 P00915 1/20 0.58
CA2 P00918 1/20 0.58
POLB P06746 1/20 0.57
ADORA3 P0DMS8 1/20 0.56
CACNA1D Q01668 2/20 0.52
CACNA1F O60840 1/20 0.52
CACNA1S Q13698 1/20 0.52
CACNA1C Q13936 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10475395 0.92 ALDH1A1 (0.78) ALDH1A1KDM4EHSD17B10HPGDTP53
SCHEMBL10475396 0.88 CACNA1B (0.74) ALDH1A1KDM4EHSD17B10HPGDTP53
SCHEMBL9064752 0.87 ADORA3 (0.74) ALDH1A1KDM4EHSD17B10HPGDTP53
SCHEMBL3022593 0.86 ADORA3 (0.59) ALDH1A1KDM4EHSD17B10HPGDMEN1
SCHEMBL24469031 0.85 ALDH1A1 (0.68) ALDH1A1KDM4EHSD17B10HPGDTP53
SCHEMBL9502874 0.82 CACNA1B (0.58) CACNA1BADORA3CACNA1DCACNA1FCACNA1S
SCHEMBL4935843 0.81 KDM4E (0.82) ALDH1A1KDM4EHSD17B10HPGDTP53
SCHEMBL9504224 0.81 KDM4E (0.61) ALDH1A1KDM4EHSD17B10HPGDTP53
SCHEMBL4624081 0.80 TP53 (0.62) ALDH1A1KDM4EHSD17B10HPGDTP53
SCHEMBL3027621 0.79 KDM4E (0.79) ALDH1A1KDM4EHSD17B10HPGDTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0458823-B1 A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA S.P.A. (IT) 1993-10-13 EP disclosed
US-5245039-A PROCESS FOR PREPARATION OF ENANTIOMERICALLY PURE POLYSUBSTITUTED 1,4-DIHYDROPYRIDINES BOEHRINGER MANNHEIM ITALIA (IT) 1993-09-14 US disclosed