SCHEMBL9503386

SCHEMBL9503386

CCOP(=O)(CC)OCc1ccc(NC(=O)C(F)(F)F)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EPHX2 P34913 3/20 0.48
NR1H4 Q96RI1 1/20 0.48
PDK1 Q15118 1/20 0.41
PDK2 Q15119 1/20 0.41
PDK3 Q15120 1/20 0.41
PDK4 Q16654 1/20 0.41
MAPT P10636 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
MEN1 O00255 1/20 0.40
ALDH1A1 P00352 1/20 0.40
RAB9A P51151 1/20 0.40
KMT2A Q03164 1/20 0.40
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA9 Q16790 1/20 0.40
S1PR4 O95977 6/20 0.39
S1PR1 P21453 6/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9500924 0.89 EPHX2 (0.47) EPHX2NR1H4PDK1PDK2PDK3
SCHEMBL5809008 0.85 EPHX2 (0.51) EPHX2NR1H4PDK1PDK2PDK3
SCHEMBL8721476 0.78 NPC1 (0.59) MEN1RAB9AKMT2ALMNA
SCHEMBL6056652 0.75 MAOB (0.49) MAPTALDH1A1RAB9AKMT2ATSHR
SCHEMBL10937278 0.75 RXRA (0.50) ALDH1A1RAB9ATSHR
SCHEMBL6056716 0.74 TSHR (0.52) ALDH1A1RAB9AKMT2ATSHRLMNA
SCHEMBL17845228 0.74 EPHX2 (0.55) EPHX2NR1H4MAPTCYP1A2CYP2C9
SCHEMBL4586654 0.73 TSHR (0.54) MAPTMEN1ALDH1A1KMT2AFPR2
SCHEMBL3196647 0.73 TSHR (0.54) MAPTALDH1A1RAB9ACA1CA2
SCHEMBL5808533 0.72 MAPT (0.39) EPHX2NR1H4PDK1PDK2PDK3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0260939-B1 MOLECULES WITH ANTIBODY COMBINING SITES THAT EXHIBIT CATALYTIC PROPERTIES SCRIPPS CLINIC AND RESEARCH FOUNDATION (US) 1993-04-28 EP disclosed
US-5126258-A Hydrolysis of polypeptides at predetermined site SCRIPPS CLINIC AND RESEARCH FOUNDATION (US) 1992-06-30 US disclosed
US-5030717-A Binding site which bind to reactant ligand, stabilization SCRIPPS CLINIC AND RESEARCH FOUNDATION (US) 1991-07-09 US disclosed
EP-0260939-A2 Molecules with antibody combining sites that exhibit catalytic properties SCRIPPS CLINIC AND RESEARCH FOUNDATION (US) 1988-03-23 EP disclosed