SCHEMBL9503589

SCHEMBL9503589

[2H]c1ccc2[nH]c(C)c(CCN)c2c1[2H]

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR6 P50406 4/20 0.54
HTR1D P28221 2/20 0.54
CYP3A4 P08684 2/20 0.54
MAPK1 P28482 2/20 0.54
CYP1A2 P05177 1/20 0.54
CYP2D6 P10635 1/20 0.54
CYP2C9 P11712 1/20 0.54
CYP2C19 P33261 1/20 0.54
HTR7 P34969 1/20 0.54
HTR3A P46098 1/20 0.54
HSD17B10 Q99714 1/20 0.54
TDP1 Q9NUW8 1/20 0.54
HTT P42858 2/20 0.47
ALDH1A1 P00352 2/20 0.47
TSHR P16473 1/20 0.47
TRPM8 Q7Z2W7 1/20 0.47
KDM4E B2RXH2 2/20 0.46
POLB P06746 1/20 0.46
NPSR1 Q6W5P4 2/20 0.45
RAD52 P43351 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1424220 0.82 ALDH1A1 (0.69) HTR6HTR1DCYP3A4MAPK1CYP1A2
SCHEMBL29415611 0.82 ALDH1A1 (0.69) HTR6HTR1DCYP3A4MAPK1CYP1A2
Hydrochloric Acid SCHEMBL273338 0.80 ALDH1A1 (0.67) HTR6HTR1DCYP3A4MAPK1CYP1A2
Cyanide SCHEMBL28575462 0.78 ALDH1A1 (0.63) HTR6HTR1DCYP3A4MAPK1CYP1A2
Oxalic Acid SCHEMBL27171318 0.74 MAPT (0.63) HTR6HTR1DCYP3A4MAPK1CYP1A2
SCHEMBL7886752 0.72 HTR1D (0.71) HTR6HTR1DCYP3A4MAPK1CYP1A2
Indole SCHEMBL28334991 0.71 ALDH1A1 (0.54) HTR6HTR1DCYP3A4MAPK1CYP1A2
SCHEMBL28750432 0.70 HTR6 (0.68) HTR6HTR1DCYP3A4MAPK1CYP1A2
SCHEMBL30619662 0.70 HTR6 (0.68) HTR6HTR1DCYP3A4MAPK1CYP1A2
SCHEMBL8244089 0.70 HTR6 (0.68) HTR6HTR1DCYP3A4MAPK1CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233413-B1 3-(2-AMINOETHYL)INDOLE AND -INDOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITHKLINE BEECHAM PHARMA GmbH (DE) 1993-05-05 EP disclosed
US-4980368-A CEREBRALVASCULAR DISORDERS; ANTIHYPOXIA AGENTS; COGNITION ACTIVATORS; SENILITY BEECHAM-WUELFING GMBH & CO. KG (DE) 1990-12-25 US disclosed
EP-0233413-A2 3-(2-Aminoethyl)indole and -indoline derivatives, processes for their preparation and pharmaceutical compositions containing them SMITHKLINE BEECHAM PHARMA GmbH (DE) 1987-08-26 EP disclosed