SCHEMBL9503716

SCHEMBL9503716

CCOC(=O)C(=O)CCCN1C(=O)c2ccccc2C1=O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.57
KMT2A Q03164 3/20 0.53
HSD17B10 Q99714 2/20 0.53
MEN1 O00255 1/20 0.53
NPSR1 Q6W5P4 2/20 0.51
TSHR P16473 2/20 0.51
MAPT P10636 1/20 0.51
MAPK1 P28482 1/20 0.51
CYP3A4 P08684 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
ACHE P22303 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
GAA P10253 1/20 0.49
HDAC8 Q9BY41 3/20 0.49
HDAC3 O15379 2/20 0.49
HDAC4 P56524 2/20 0.49
HDAC1 Q13547 2/20 0.49
HDAC7 Q8WUI4 2/20 0.49
HDAC2 Q92769 2/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7852944 0.91 HPGD (0.53) ALDH1A1KMT2AMEN1TSHRMAPT
SCHEMBL7424373 0.85 KMT2A (0.63) ALDH1A1KMT2AHSD17B10MEN1NPSR1
SCHEMBL7260269 0.85 ALDH1A1 (0.54) ALDH1A1KMT2AHSD17B10MEN1NPSR1
SCHEMBL1233999 0.83 KMT2A (0.51) ALDH1A1KMT2AMEN1MAPTGAA
SCHEMBL398553 0.82 ALDH1A1 (0.59) ALDH1A1KMT2AMEN1NPSR1MAPT
SCHEMBL31440149 0.82 ALDH1A1 (0.59) ALDH1A1KMT2AMEN1NPSR1MAPT
SCHEMBL15679600 0.81 ALDH1A1 (0.55) ALDH1A1KMT2AHSD17B10MEN1NPSR1
SCHEMBL9798967 0.81 ALDH1A1 (0.58) ALDH1A1KMT2AHSD17B10MEN1NPSR1
SCHEMBL7589770 0.80 HDAC8 (0.59) ALDH1A1KMT2AHSD17B10MEN1TSHR
SCHEMBL7549194 0.80 HDAC8 (0.59) ALDH1A1KMT2AHSD17B10MEN1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0233413-B1 3-(2-AMINOETHYL)INDOLE AND -INDOLINE DERIVATIVES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM SMITHKLINE BEECHAM PHARMA GmbH (DE) 1993-05-05 EP disclosed
US-4980368-A CEREBRALVASCULAR DISORDERS; ANTIHYPOXIA AGENTS; COGNITION ACTIVATORS; SENILITY BEECHAM-WUELFING GMBH & CO. KG (DE) 1990-12-25 US disclosed
EP-0233413-A2 3-(2-Aminoethyl)indole and -indoline derivatives, processes for their preparation and pharmaceutical compositions containing them SMITHKLINE BEECHAM PHARMA GmbH (DE) 1987-08-26 EP disclosed