SCHEMBL9507172

SCHEMBL9507172

CC1CC1(Cl)Cl.O=C(O)Cl

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
APLNR P35414 1/20 0.36
GRM2 Q14416 3/20 0.33
GRM3 Q14832 3/20 0.33
CYP2C19 P33261 1/20 0.33
GAA P10253 2/20 0.32
THRB P10828 2/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 2/20 0.32
TSHR P16473 2/20 0.32
CYP2C9 P11712 2/20 0.32
BLM P54132 1/20 0.32
PPARA Q07869 1/20 0.32
GRM6 O15303 2/20 0.30
EPHX1 P07099 1/20 0.30
CYP1A2 P05177 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Bicarbonate SCHEMBL10606286 0.91 APLNR (0.38) APLNRGRM2GRM3CYP2C19LMNA
Bicarbonate SCHEMBL4003894 0.91 APLNR (0.38) APLNRGRM2GRM3CYP2C19LMNA
SCHEMBL6714807 0.91 GAA (0.38) APLNRGRM2GRM3GAATHRB
Cyclopentane SCHEMBL10864965 0.86 APLNR (0.35) APLNRCYP2C19LMNATSHRCYP2C9
SCHEMBL9485514 0.83 APLNR (0.33) APLNRGRM2GRM3CYP2C19GAA
SCHEMBL18534475 0.80
SCHEMBL111139 0.80
SCHEMBL13783354 0.80
SCHEMBL1744322 0.80 APLNR (0.35) APLNRGRM2GRM3CYP2C19
Formic Acid SCHEMBL27756908 0.77

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0398059-B1 CYCLOPROPANOYLAMINOACID AMIDE DERIVATIVES BAYER AG (DE) 1993-08-25 EP disclosed
EP-0398059-A1 Cyclopropanoylaminoacid amide derivatives BAYER AG (DE) 1990-11-22 EP disclosed
EP-0195201-B1 PROCESS FOR THE PREPARATION OF N-ACYL-2,3-DEHYDRO CARBOXYLIC ESTERS Degussa Aktiengesellschaft (DE) 1990-05-23 EP disclosed
EP-0257448-A2 Optically active cyclopropanecarboxamides NIHON BAYER AGROCHEM K.K. (JP) 1988-03-02 EP disclosed
EP-0195201-A2 Process for the preparation of N-acyl-2,3-dehydro carboxylic esters Degussa Aktiengesellschaft (DE) 1986-09-24 EP disclosed
EP-0042107-B1 DIHYDROPYRIDAZINONES, PROCESSES FOR THEIR PREPARATION AND PHARMACEUTICAL COMPOSITIONS CONTAINING THESE COMPOUNDS BASF Aktiengesellschaft (DE) 1985-04-03 EP disclosed
EP-0042107-A1 Dihydropyridazinones, processes for their preparation and pharmaceutical compositions containing these compounds BASF Aktiengesellschaft (DE) 1981-12-23 EP disclosed