SCHEMBL9507469

SCHEMBL9507469

COC(=O)/C=C/c1cc(C(F)(F)F)ccc1CCCCCCCCc1ccccc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYSLTR2 Q9NS75 1/20 0.48
CYSLTR1 Q9Y271 1/20 0.48
AKR1B10 O60218 2/20 0.43
AKR1B1 P15121 2/20 0.43
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
GAA P10253 1/20 0.41
MAPT P10636 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC8 Q9BY41 1/20 0.41
ALOX5 P09917 2/20 0.40
NR1H4 Q96RI1 1/20 0.40
NOS3 P29474 1/20 0.40
NOS1 P29475 1/20 0.40
NOS2 P35228 1/20 0.40
PLK1 P53350 1/20 0.40
RXRA P19793 1/20 0.40
NR1H2 P55055 1/20 0.40
NR1H3 Q13133 1/20 0.40
ASAH1 Q13510 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9507472 1.00 CYSLTR2 (0.48) CYSLTR2CYSLTR1AKR1B10AKR1B1ALDH1A1
SCHEMBL9560089 0.89 RXRA (0.49) CYSLTR2CYSLTR1AKR1B10AKR1B1ALDH1A1
SCHEMBL9560090 0.89 RXRA (0.49) CYSLTR2CYSLTR1AKR1B10AKR1B1ALDH1A1
SCHEMBL10424229 0.88 CYSLTR2 (0.53) CYSLTR2CYSLTR1MAPTHDAC1HDAC8
SCHEMBL10424230 0.88 CYSLTR2 (0.53) CYSLTR2CYSLTR1MAPTHDAC1HDAC8
SCHEMBL9481085 0.79 CYSLTR2 (0.52) CYSLTR2CYSLTR1MAPTHDAC1HDAC8
SCHEMBL9721103 0.78 CYSLTR2 (0.44) CYSLTR2CYSLTR1ALDH1A1LMNAMAPT
SCHEMBL9721098 0.78 CYSLTR2 (0.44) CYSLTR2CYSLTR1ALDH1A1LMNAMAPT
SCHEMBL9493070 0.76 ALDH1A1 (0.51) ALDH1A1LMNAGAAMAPT
SCHEMBL9493078 0.76 ALDH1A1 (0.51) ALDH1A1LMNAGAAMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0375348-B1 LEUKOTRIENE ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1993-06-23 EP disclosed
US-4954513-A Leukotriene antagonists SMITHKLINE BEECHAM CORPORATION (US) 1990-09-04 US disclosed