SCHEMBL9507496

SCHEMBL9507496

COc1cccc(CN(C)C)c1SCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 2/20 0.46
SLC6A4 P31645 5/20 0.46
SLC6A2 P23975 4/20 0.46
SLC6A3 Q01959 3/20 0.46
RAB9A P51151 2/20 0.42
L3MBTL1 Q9Y468 1/20 0.42
CTSB P07858 1/20 0.42
BCHE P06276 2/20 0.41
EGFR P00533 1/20 0.41
ALDH1A1 P00352 3/20 0.41
TSHR P16473 2/20 0.41
MEN1 O00255 1/20 0.40
CRHBP P24387 1/20 0.40
KMT2A Q03164 1/20 0.40
CRHR2 Q13324 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
TP53 P04637 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9510856 0.82 RAB9A (0.44) RAB9AL3MBTL1CTSBBCHEEGFR
SCHEMBL5345977 0.82 SLC6A4 (0.47) HTR7SLC6A4SLC6A2SLC6A3HTR2A
SCHEMBL5340091 0.80 SLC6A4 (0.50) HTR7SLC6A4SLC6A2SLC6A3HTR2A
SCHEMBL10701574 0.79 SLC6A4 (0.48) HTR7SLC6A4SLC6A2SLC6A3TSHR
SCHEMBL31172708 0.76 RAB9A (0.46) SLC6A4RAB9AL3MBTL1CTSBEGFR
SCHEMBL31172667 0.76 TP53 (0.48) RAB9AL3MBTL1CTSBEGFRALDH1A1
SCHEMBL31172733 0.75 NR2E3 (0.49) RAB9AL3MBTL1CTSBEGFRALDH1A1
SCHEMBL735118 0.74 SLC6A4 (0.68) HTR7SLC6A4SLC6A2SLC6A3MEN1
SCHEMBL31172632 0.74 RAB9A (0.44) SLC6A4RAB9AL3MBTL1CTSBEGFR
SCHEMBL31510902 0.74 HTR1A (0.46) RAB9AL3MBTL1CTSBEGFRALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0358305-B1 MERCAPTO-PHENYLALCANOYLAMINO ACID AMIDES, THEIR PREPARATION AND THEIR USE AS COLLAGENASE INHIBITORS BEECHAM GROUP PLC (GB) 1993-08-25 EP disclosed
US-5124322-A Antiarthritic agents BEECHAM GROUP P.L.C. (GB) 1992-06-23 US disclosed
EP-0358305-A1 Mercapto-phenylalcanoylamino acid amides, their preparation and their use as collagenase inhibitors BEECHAM GROUP PLC (GB) 1990-03-14 EP disclosed