SCHEMBL9509427

SCHEMBL9509427

CCCOc1ccc(C#Cc2ccc([C@H]3CC[C@H](C)CC3)cc2)c(F)c1F

nearest known ligand 0.35

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.35
ACACB O00763 9/20 0.33
RAB9A P51151 1/20 0.32
HRH3 Q9Y5N1 1/20 0.32
PDE4A P27815 2/20 0.31
HTR2A P28223 2/20 0.31
CHRM1 P11229 1/20 0.31
MCHR1 Q99705 1/20 0.31
HTR2C P28335 2/20 0.30
HTR2B P41595 2/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9512298 0.94 RAB9A (0.38) ESR2ACACBRAB9AHRH3PDE4A
SCHEMBL9509280 0.93 RAB9A (0.35) ESR2ACACBRAB9AHRH3
SCHEMBL21165799 0.92 ESR2 (0.37) ESR2ACACBHRH3HTR2ACHRM1
SCHEMBL9511367 0.92 ESR2 (0.37) ESR2ACACBHRH3HTR2ACHRM1
SCHEMBL9512338 0.90 ACACB (0.34) ACACBPDE4A
SCHEMBL9508834 0.89 CYP2C9 (0.39) ESR2ACACBPDE4A
SCHEMBL9510141 0.87 ACACB (0.33) ACACBRAB9AHRH3
SCHEMBL9508734 0.86 ACACB (0.33) ACACBRAB9AHRH3
SCHEMBL10515991 0.86 CYP2C9 (0.31)
SCHEMBL9512361 0.85 SPHK1 (0.33) ACACBRAB9AHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308438-B1 LIQUID CRYSTAL PHASE CONTAINING TOLANES MERCK PATENT GmbH (DE) 1993-09-29 EP disclosed