SCHEMBL9511367

SCHEMBL9511367

CCOc1ccc(C#Cc2ccc([C@H]3CC[C@H](C)CC3)cc2)c(F)c1F

nearest known ligand 0.37

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 1/20 0.37
KDM1A O60341 2/20 0.35
HRH3 Q9Y5N1 1/20 0.31
ALDH1A1 P00352 1/20 0.31
ACACB O00763 2/20 0.31
MEN1 O00255 1/20 0.30
KMT2A Q03164 1/20 0.30
CHRM1 P11229 1/20 0.30
HTR2A P28223 1/20 0.30
MCHR1 Q99705 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21165799 1.00 ESR2 (0.37) ESR2KDM1AHRH3ALDH1A1ACACB
SCHEMBL9509427 0.92 ESR2 (0.35) ESR2HRH3ACACBCHRM1HTR2A
SCHEMBL9512298 0.91 RAB9A (0.38) ESR2HRH3ACACBCHRM1HTR2A
SCHEMBL9509280 0.90 RAB9A (0.35) ESR2HRH3ALDH1A1ACACB
SCHEMBL9509015 0.89 ACACB (0.38) KDM1AACACB
SCHEMBL21165795 0.89 KDM1A (0.36) KDM1AHRH3ALDH1A1MEN1KMT2A
SCHEMBL91984 0.88 ESR2 (0.39) ESR2KDM1A
SCHEMBL12230852 0.88 ESR2 (0.39) ESR2KDM1A
SCHEMBL9512291 0.88 ESR2 (0.39) ESR2KDM1A
SCHEMBL21165797 0.87 CYP2C9 (0.41) ESR2KDM1AALDH1A1ACACBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0308438-B1 LIQUID CRYSTAL PHASE CONTAINING TOLANES MERCK PATENT GmbH (DE) 1993-09-29 EP claimed
EP-0308438-B1 LIQUID CRYSTAL PHASE CONTAINING TOLANES MERCK PATENT GmbH (DE) 1993-09-29 EP disclosed