SCHEMBL9510455

SCHEMBL9510455

COc1c(C)cc(C(=O)CCCCCBr)c(C)c1OC

nearest known ligand 0.38

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.38
HDAC8 Q9BY41 3/20 0.35
HDAC1 Q13547 3/20 0.35
MAPK1 P28482 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
LMNA P02545 1/20 0.35
ALDH1A1 P00352 1/20 0.34
PDE4B Q07343 1/20 0.34
POLB P06746 1/20 0.34
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27200193 0.80 HDAC8 (0.41) HDAC8HDAC1MAPK1SMN1; SMN2LMNA
SCHEMBL9972448 0.79 HDAC8 (0.43) HTTHDAC8HDAC1PDE4BTHRA
SCHEMBL27200200 0.77 CTNNB1 (0.43) HTTHDAC8HDAC1PDE4BPOLB
SCHEMBL24783614 0.76 PLA2G2A (0.39) HDAC8HDAC1MAPK1SMN1; SMN2LMNA
SCHEMBL9508047 0.76 PLA2G2A (0.39) HDAC8HDAC1MAPK1SMN1; SMN2LMNA
SCHEMBL9972449 0.74 HTT (0.44) HTTLMNAALDH1A1
SCHEMBL8711802 0.73 PLAU (0.41) HTTHDAC8HDAC1MAPK1SMN1; SMN2
SCHEMBL23534095 0.73 POLB (0.41) HDAC8HDAC1MAPK1SMN1; SMN2ALDH1A1
SCHEMBL29767827 0.73 POLB (0.41) HDAC8HDAC1MAPK1SMN1; SMN2ALDH1A1
SCHEMBL1441802 0.73 KMT2A (0.49) HDAC8HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0310126-B1 DERIVATIVES OF PYROCATECHOL-CARBOXYLIC ACID, THEIR PREPARATION AND USE AS ACTIVE INGREDIENTS IN MEDICINES F. HOFFMANN-LA ROCHE AG (CH) 1993-08-18 EP disclosed
US-5191108-A Lipoxygenase inhibitors, antiinflammatory agents HOFFMANN-LA ROCHE INC. (US) 1993-03-02 US disclosed
US-5025036-A Antiinflammatory agents, gastrointestinal, cardiovascular and skin disorders HOFFMANN-LA ROCHE INC. (US) 1991-06-18 US disclosed
US-4937373-A Substituted naphthalene carboxylic acids HOFFMANN-LA ROCHE INC. (US) 1990-06-26 US disclosed
EP-0310126-A2 Derivatives of pyrocatechol-carboxylic acid, their preparation and use as active ingredients in medicines F. HOFFMANN-LA ROCHE AG (CH) 1989-04-05 EP disclosed