SCHEMBL9513345

SCHEMBL9513345

O=C(c1ccc(Cl)cc1)N1CCN(CCc2ccc(F)cc2)CC1

nearest known ligand 0.78

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.73
HSP90AA1 P07900 1/20 0.61
MEN1 O00255 1/20 0.60
KMT2A Q03164 1/20 0.60
KCNH2 Q12809 1/20 0.60
PRKAA2 P54646 1/20 0.60
GPR183 P32249 1/20 0.59
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.57
MAPT P10636 1/20 0.57

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9513181 1.00 THRB (0.73) THRBHSP90AA1MEN1KMT2AKCNH2
Hydrochloric Acid SCHEMBL9516740 0.99 THRB (0.71) THRBHSP90AA1MEN1KMT2AKCNH2
SCHEMBL9513241 0.93 THRB (0.82) THRBMEN1KMT2AKCNH2GPR183
SCHEMBL9513154 0.93 MEN1 (0.68) THRBMEN1KMT2AKCNH2PRKAA2
SCHEMBL10901582 0.88 THRB (0.74) THRBMEN1KMT2AKCNH2GPR183
SCHEMBL9512997 0.87 THRB (0.73) THRBMEN1KMT2AKCNH2GPR183
SCHEMBL9136775 0.87 THRB (0.73) THRBMEN1KMT2AKCNH2GPR183
SCHEMBL9426176 0.87 MEN1 (0.60) THRBMEN1KMT2AKCNH2PRKAA2
SCHEMBL10898714 0.87 THRB (0.73) THRBMEN1KMT2AKCNH2GPR183
SCHEMBL9515645 0.86 THRB (0.72) THRBMEN1KMT2AKCNH2PRKAA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0250361-B1 Disubstituted piperazines CIBA GEIGY AG (CH) 1993-12-08 EP claimed
EP-0250361-A2 Disubstituted piperazines CIBA-GEIGY AG (CH) 1987-12-23 EP claimed
US-4804661-A ANALGESICS CIBA-GEIGY CORPORATION (US) 1989-02-14 US disclosed