SCHEMBL9515645

SCHEMBL9515645

O=C(c1ccc(C(F)(F)F)cc1)N1CCN(CCc2ccc(Cl)cc2)CC1

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
THRB P10828 2/20 0.72
SIGMAR1 Q99720 1/20 0.62
PRKAB2 O43741 4/20 0.61
PRKAG1 P54619 4/20 0.61
PRKAA2 P54646 4/20 0.61
PRKAA1 Q13131 4/20 0.61
PRKAG3 Q9UGI9 4/20 0.61
PRKAG2 Q9UGJ0 4/20 0.61
PRKAB1 Q9Y478 4/20 0.61
MGLL Q99685 1/20 0.58
MEN1 O00255 3/20 0.56
KMT2A Q03164 3/20 0.56
KCNH2 Q12809 1/20 0.56
GPR183 P32249 1/20 0.55
KDM4E B2RXH2 1/20 0.54
ALDH1A1 P00352 1/20 0.54
MAPT P10636 1/20 0.54
LSS P48449 1/20 0.54
LMNA P02545 1/20 0.54
HPGD P15428 1/20 0.53

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9514281 0.99 THRB (0.70) THRBSIGMAR1PRKAB2PRKAG1PRKAA2
SCHEMBL9513241 0.90 THRB (0.82) THRBMEN1KMT2AKCNH2GPR183
SCHEMBL9514284 0.86 LMNA (0.61) THRBMGLLMEN1KMT2AKCNH2
SCHEMBL9513181 0.86 THRB (0.73) THRBPRKAA2MEN1KMT2AKCNH2
SCHEMBL9513345 0.86 THRB (0.73) THRBPRKAA2MEN1KMT2AKCNH2
Hydrochloric Acid SCHEMBL9514278 0.85 LMNA (0.60) THRBPRKAB2PRKAG1PRKAA2PRKAA1
Hydrochloric Acid SCHEMBL9516740 0.85 THRB (0.71) THRBPRKAA2MEN1KMT2AKCNH2
SCHEMBL10901582 0.85 THRB (0.74) THRBSIGMAR1MEN1KMT2AKCNH2
SCHEMBL10898714 0.84 THRB (0.73) THRBMEN1KMT2AKCNH2GPR183
SCHEMBL9512997 0.84 THRB (0.73) THRBMGLLMEN1KMT2AKCNH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0250361-B1 Disubstituted piperazines CIBA GEIGY AG (CH) 1993-12-08 EP claimed
EP-0250361-A2 Disubstituted piperazines CIBA-GEIGY AG (CH) 1987-12-23 EP claimed