SCHEMBL9514911

SCHEMBL9514911

ClCCON=C(c1ccccc1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBXA2R P21731 9/20 0.48
TBXAS1 P24557 5/20 0.48
ALDH1A1 P00352 3/20 0.46
CYP1A2 P05177 2/20 0.46
CYP2D6 P10635 2/20 0.46
CYP2C9 P11712 2/20 0.46
CYP2C19 P33261 2/20 0.46
CYP3A4 P08684 1/20 0.46
HPGD P15428 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
KDM4E B2RXH2 2/20 0.43
LMNA P02545 2/20 0.43
BLM P54132 2/20 0.43
PMP22 Q01453 2/20 0.43
KMT2A Q03164 2/20 0.43
TP53 P04637 1/20 0.43
ALOX12 P18054 1/20 0.43
MAPK1 P28482 1/20 0.43
ESR1 P03372 1/20 0.43
PPARG P37231 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22946578 0.80 PPARG (0.59) TBXA2RTBXAS1ALDH1A1CYP1A2CYP2D6
SCHEMBL27835726 0.78 PPARG (0.48) TBXA2RTBXAS1ALDH1A1CYP1A2CYP2D6
SCHEMBL3883360 0.78 TBXA2R (0.54) TBXA2RTBXAS1ESR1
SCHEMBL14596992 0.77 ALDH1A1 (0.50) TBXA2RTBXAS1ALDH1A1CYP1A2CYP2D6
SCHEMBL1115510 0.76 HTR1D (0.47) TBXA2RTBXAS1ALDH1A1CYP1A2CYP2D6
SCHEMBL3884214 0.76 TBXA2R (0.44) TBXA2RTBXAS1ALDH1A1CYP1A2CYP2D6
SCHEMBL13351521 0.75 ALDH1A1 (0.49) TBXA2RTBXAS1ALDH1A1CYP1A2CYP2D6
SCHEMBL4259732 0.75 ALDH1A1 (0.49) TBXA2RTBXAS1ALDH1A1CYP1A2CYP2D6
SCHEMBL10892857 0.74 TBXA2R (0.74) TBXA2RTBXAS1PPARA
SCHEMBL10452205 0.73 SMN1; SMN2 (0.49) TBXA2RTBXAS1ALDH1A1CYP1A2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5231106-A Nervous sytem disorders; blocking og gamma aminobutyric acid NOVO NORDISK A/S (DK) 1993-07-27 US disclosed
US-5229404-A Inhibitors of gamma-aminobutyric acid re-uptake, antiepileptic agents NOVO NORDISK A/S (DK) 1993-07-20 US disclosed
US-5214054-A Gamma-aminobutyric acid re-uptake inhibitors, antiepileptic, analgesics, anxiolytics NOVO NORDISK A/S (DK) 1993-05-25 US disclosed
US-5039685-A Nervous system disorders NOVO NORDISK A/S (DK) 1991-08-13 US disclosed