SCHEMBL4259732

SCHEMBL4259732

[CH2]CON=C(c1ccccc1)c1ccccc1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
CYP1A2 P05177 2/20 0.49
CYP2D6 P10635 2/20 0.49
CYP2C9 P11712 2/20 0.49
CYP2C19 P33261 2/20 0.49
CYP3A4 P08684 1/20 0.49
HPGD P15428 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
LMNA P02545 3/20 0.44
MAPK1 P28482 2/20 0.44
HTT P42858 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
TBXA2R P21731 9/20 0.43
TBXAS1 P24557 5/20 0.43
KDM4E B2RXH2 2/20 0.42
BLM P54132 2/20 0.42
PMP22 Q01453 2/20 0.42
KMT2A Q03164 2/20 0.42
TP53 P04637 1/20 0.42
ALOX12 P18054 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14596992 0.80 ALDH1A1 (0.50) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL9362227 0.79 LMNA (0.47) SMN1; SMN2LMNAKMT2AESR1
SCHEMBL13351521 0.78 ALDH1A1 (0.49) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL10452205 0.77 SMN1; SMN2 (0.49) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
Hydrochloric Acid SCHEMBL27649130 0.75 SMN1; SMN2 (0.47) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL22946578 0.75 PPARG (0.59) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL9514911 0.75 TBXA2R (0.48) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL8613026 0.75 TBXA2R (0.51) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL27835726 0.74 PPARG (0.48) ALDH1A1CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL3883360 0.74 TBXA2R (0.54) TBXA2RTBXAS1ESR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009042723-A1 TRANSGENIC MICE EXPRESSING HYPERSENSITIVE NICOTINIC RECEPTORS CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2009-04-02 WO disclosed
EP-1951212-A2 COMPOSITIONS AND METHODS FOR INCREASING INSULIN SENSITIVITY Orexigen Therapeutics, Inc. (US) 2008-08-06 EP disclosed
WO-2007067341-A2 COMPOSITIONS AND METHODS FOR INCREASING INSULIN SENSITIVITY OREXIGEN THERAPEUTICS, INC. (US) 2007-06-14 WO disclosed