SCHEMBL9514912

SCHEMBL9514912

CCCCCNCc1ccc2[nH]cnc(=O)c2c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.46
CYP2D6 P10635 3/20 0.46
CYP2C19 P33261 3/20 0.46
HRH4 Q9H3N8 1/20 0.46
HRH3 Q9Y5N1 1/20 0.46
LMNA P02545 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.43
EPHX1 P07099 1/20 0.41
S1PR2 O95136 2/20 0.39
S1PR1 P21453 2/20 0.39
S1PR3 Q99500 2/20 0.39
LPAR2 Q9HBW0 2/20 0.39
KDM4E B2RXH2 1/20 0.39
PARP1 P09874 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9514916 0.80 IP6K1 (0.52) HRH4HRH3EPHX1PARP1
SCHEMBL27797161 0.68 TNKS2 (0.48) CYP1A2CYP2D6CYP2C19HRH4HRH3
SCHEMBL10747074 0.67 HRH4 (0.84) CYP1A2CYP2D6CYP2C19HRH4HRH3
SCHEMBL9259496 0.67 HRH4 (0.84) CYP1A2CYP2D6CYP2C19HRH4HRH3
SCHEMBL10748421 0.67 HRH4 (0.84) CYP1A2CYP2D6CYP2C19HRH4HRH3
SCHEMBL9637156 0.67 HRH4 (0.84) CYP1A2CYP2D6CYP2C19HRH4HRH3
SCHEMBL1507612 0.67 PARP1 (0.54) LMNASMN1; SMN2KDM4EPARP1
SCHEMBL1507706 0.66 TYMS (0.41) CYP1A2SMN1; SMN2KDM4EPARP1
SCHEMBL1584889 0.65 PIM1 (0.56) CYP1A2LMNASMN1; SMN2
SCHEMBL9257479 0.65 CYP1A2 (0.76) CYP1A2CYP2D6CYP2C19HRH4HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0284338-B1 Anti-tumour agents ICI PLC (GB) 1993-12-22 EP disclosed