SCHEMBL9515018

SCHEMBL9515018

CC(C)(C)OC(=O)NC1Cc2ccc3ccccc3c2CC1=O

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 1/20 0.52
EPHX2 P34913 1/20 0.41
GAA P10253 2/20 0.40
NFKB1 P19838 2/20 0.39
NFKB2 Q00653 2/20 0.39
RELA Q04206 2/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
NPC1 O15118 1/20 0.38
RAB9A P51151 1/20 0.38
ATM Q13315 1/20 0.37
CCKBR P32239 1/20 0.37
KDM1A O60341 1/20 0.37
MAOB P27338 1/20 0.37
PDE10A Q9Y233 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9513864 0.79 EPHX2 (0.51) ANPEPEPHX2GAANFKB1NFKB2
SCHEMBL9515367 0.79 EPHX2 (0.41) ANPEPEPHX2GAANFKB1NFKB2
SCHEMBL9515374 0.79 EPHX2 (0.41) ANPEPEPHX2GAANFKB1NFKB2
SCHEMBL9515381 0.79 EPHX2 (0.41) ANPEPEPHX2GAANFKB1NFKB2
SCHEMBL9515379 0.78 EPHX2 (0.50) ANPEPEPHX2GAANFKB1NFKB2
SCHEMBL1718456 0.71 DRD2 (0.48) ANPEPEPHX2GAANFKB1NFKB2
SCHEMBL9513876 0.69 ANPEP (1.00) ANPEP
SCHEMBL10446636 0.69 EPHX2 (0.49) EPHX2GAANFKB1NFKB2RELA
SCHEMBL26518868 0.69 GAA (0.38) EPHX2GAANFKB1NFKB2RELA
Isoamylamine SCHEMBL10446310 0.69 EPHX2 (0.44) EPHX2GAANFKB1NFKB2RELA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0378456-B1 TETRALIN DERIVATIVES MERRELL DOW PHARMACEUTICALS INC. (US) 1993-09-15 EP disclosed
US-5106861-A Method of using certain tetralin derivatives to produce analgesic relief MERRELL DOW PHARMACEUTICALS INC. (US) 1992-04-21 US disclosed
US-5041673-A Aminopeptidase inhibitors, immunomodulators, analgesics MERRELL DOW PHARMACEUTICALS INC. (US) 1991-08-20 US disclosed
EP-0378456-A1 Tetralin derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1990-07-18 EP disclosed