SCHEMBL9515925

SCHEMBL9515925

O=P(O)(O)C=CCc1ncc2[nH]cnc2n1

nearest known ligand 0.41

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
KDM4E B2RXH2 1/20 0.41
RXFP1 Q9HBX9 1/20 0.40
CDK2 P24941 2/20 0.34
PAK1 Q13153 1/20 0.33
CCNT1 O60563 1/20 0.32
CDK1 P06493 1/20 0.32
CCNB1 P14635 1/20 0.32
CDK7 P50613 1/20 0.32
CDK9 P50750 1/20 0.32
CCNH P51946 1/20 0.32
POLA1 P09884 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL609326 0.81 ALDH1A1 (0.46) ALDH1A1KDM4ERXFP1CDK2PAK1
SCHEMBL460357 0.81 ALDH1A1 (0.36) ALDH1A1KDM4ERXFP1CDK2
SCHEMBL11498403 0.78 ALDH1A1 (0.50) ALDH1A1KDM4ERXFP1CDK2PAK1
SCHEMBL9516025 0.78
SCHEMBL1079075 0.74 ALDH1A1 (0.49) ALDH1A1KDM4ERXFP1CDK2PAK1
SCHEMBL8607904 0.72 ALDH1A1 (0.41) ALDH1A1KDM4ERXFP1CDK2PAK1
SCHEMBL3044447 0.72 ALDH1A1 (0.41) ALDH1A1KDM4ERXFP1CDK2PAK1
SCHEMBL3054589 0.71 ALDH1A1 (0.40) ALDH1A1KDM4ERXFP1CDK2PAK1
SCHEMBL31618832 0.70 ALDH1A1 (0.47) ALDH1A1KDM4ERXFP1CDK2PAK1
SCHEMBL8708640 0.69 ALDH1A1 (0.38) ALDH1A1KDM4ERXFP1CDK2PAK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0338887-B1 Phosphonoalkylpurine derivatives MERRELL DOW PHARMA (US) 1993-12-08 EP disclosed
EP-0338887-B1 Phosphonoalkylpurine derivatives MERRELL DOW PHARMA (US) 1993-12-08 EP disclosed
US-4988680-A Phosphorylase inhibitors, immuno suppressants, parasiticides, antileukemia agents MERRELL DOW PHARMACEUTICALS INC. (US) 1991-01-29 US disclosed
US-4988680-A Phosphorylase inhibitors, immuno suppressants, parasiticides, antileukemia agents MERRELL DOW PHARMACEUTICALS INC. (US) 1991-01-29 US disclosed
EP-0338887-A1 Phosphonoalkylpurine derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1989-10-25 EP disclosed
EP-0338168-A1 Phosphonoalkylpurine derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1989-10-25 EP disclosed
EP-0338887-A1 Phosphonoalkylpurine derivatives MERRELL DOW PHARMACEUTICALS INC. (US) 1989-10-25 EP disclosed