SCHEMBL9518571

SCHEMBL9518571

COC(=O)CC(=O)CON=C(c1ccc(OC)cc1)c1ccc(OC)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.46
L3MBTL1 Q9Y468 2/20 0.46
GAA P10253 1/20 0.46
KMT2A Q03164 1/20 0.46
CA1 P00915 5/20 0.45
CA2 P00918 5/20 0.45
LMNA P02545 2/20 0.43
CES2 O00748 1/20 0.43
CES1 P23141 1/20 0.43
PLK1 P53350 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
GSK3B P49841 1/20 0.41
HDAC3 O15379 1/20 0.41
HDAC4 P56524 1/20 0.41
HDAC1 Q13547 1/20 0.41
HDAC7 Q8WUI4 1/20 0.41
HDAC2 Q92769 1/20 0.41
HDAC10 Q969S8 1/20 0.41
HDAC11 Q96DB2 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9516306 0.89 KMT2A (0.45) MAPTL3MBTL1GAAKMT2ACA1
SCHEMBL9518576 0.85 TBXAS1 (0.47) MAPTL3MBTL1GAAKMT2ACES2
SCHEMBL9520420 0.85 MAPT (0.43) MAPTL3MBTL1GAAKMT2ACA1
SCHEMBL11527620 0.81 CA1 (0.52) MAPTL3MBTL1GAAKMT2ACA1
SCHEMBL11524689 0.79 HDAC3 (0.47) MAPTL3MBTL1GAAKMT2ACES2
SCHEMBL9520361 0.78 PLA2G4B (0.47) MAPTL3MBTL1GAALMNAPLK1
SCHEMBL9516891 0.76 CA1 (0.42) MAPTL3MBTL1GAAKMT2ACA1
SCHEMBL9516341 0.75 ALDH1A1 (0.43) MAPTL3MBTL1GAAKMT2ACA1
SCHEMBL9516296 0.73 MAPT (0.48) MAPTGAAKMT2ALMNACES2
SCHEMBL17295084 0.72 ALDH1A1 (0.64) MAPTKMT2ACA1CA2LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5206403-A Diphenylethylene derivatives, pharmaceutical compositions containing same and treatment methods EISAI CO., LTD. (JP) 1993-04-27 US disclosed
EP-0346943-B1 DIPHENYL-METHANE DERIVATIVE, PHARMACEUTICAL COMPOSITION AND USE Eisai Co., Ltd. (JP) 1993-02-17 EP disclosed
US-5182301-A Anticoagulants EISAI CO., LTD. (JP) 1993-01-26 US disclosed
EP-0479332-A2 Diphenyl-methane derivative, pharmaceutical composition and use Eisai Co., Ltd. (JP) 1992-04-08 EP disclosed
US-5103010-A DIPHENYLETHYLENE DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING SAME AND TREATMENT METHOD EISAI CO., LTD. (JP) 1992-04-07 US disclosed
EP-0478001-A1 Benzophenone oxime derivatives, pharmaceutical compositions and use Eisai Co., Ltd. (JP) 1992-04-01 EP disclosed
US-5034418-A Anticoagulants EISAI CO., LTD. (JP) 1991-07-23 US disclosed
US-4978767-A ANTICOAGULANTS EISAI CO., LTD. (JP) 1990-12-18 US disclosed
US-4886834-A ANTICOAGULANTS EISAI CO., LTD. (JP) 1989-12-12 US disclosed