SCHEMBL9518810

SCHEMBL9518810

CN1CCC(c2c[nH]c3ccc(CCNS(C)(=O)=O)cc23)CC1

nearest known ligand 0.71

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 13/20 0.71
HTR1B P28222 13/20 0.71
HTR1A P08908 2/20 0.71
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
THPO P40225 1/20 0.55
HTR1F P30939 2/20 0.53
APP P05067 1/20 0.53
HTR6 P50406 3/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9773080 0.99 HTR1D (0.70) HTR1DHTR1BHTR1ACYP1A2CYP3A4
SCHEMBL9527477 0.86 HTR1D (0.78) HTR1DHTR1BHTR1ACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9874795 0.85 HTR1D (0.77) HTR1DHTR1BHTR1ACYP1A2CYP3A4
SCHEMBL9874164 0.83 HTR1D (0.68) HTR1DHTR1BHTR1ACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL9265610 0.83 HTR1D (0.59) HTR1DHTR1BHTR1ACYP1A2CYP3A4
Naratriptan SCHEMBL68753 0.83 HTR1D (1.00) HTR1DHTR1BHTR1ACYP1A2CYP3A4
Naratriptan SCHEMBL29403931 0.83 HTR1D (1.00) HTR1DHTR1BHTR1ACYP1A2CYP3A4
SCHEMBL23394791 0.83 HTR1D (0.77) HTR1DHTR1BHTR1ACYP1A2CYP3A4
SCHEMBL3222849 0.83 HTR1D (0.77) HTR1DHTR1BHTR1ACYP1A2CYP3A4
SCHEMBL4541547 0.83 HTR1D (0.77) HTR1DHTR1BHTR1ACYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5036078-A And of chronic paroxysmal hemicrania GLAXO GROUP LIMITED (GB) 1991-07-30 US claimed
EP-0354777-B1 3-(4-PIPERIDINE)-5-(2-SULFONYLAMINOETHYL) INDOLE DERIVATIVES GLAXO GROUP LIMITED (GB) 1993-08-04 EP disclosed
US-5036078-A And of chronic paroxysmal hemicrania GLAXO GROUP LIMITED (GB) 1991-07-30 US disclosed
EP-0354777-A2 3-(4-Piperidine)-5-(2-sulfonylaminoethyl) indole derivatives GLAXO GROUP LIMITED (GB) 1990-02-14 EP disclosed