SCHEMBL9519685

SCHEMBL9519685

CCNC(=O)c1cccc(S(=O)(=O)NC(=O)c2ccc(CO)nc2)c1

nearest known ligand 0.48

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASP3 P42574 4/20 0.48
P4HTM Q9NXG6 3/20 0.47
SMN1; SMN2 Q16637 1/20 0.47
PTGS2 P35354 2/20 0.42
HTT P42858 1/20 0.41
NAMPT P43490 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
PTGS1 P23219 1/20 0.41
EGFR P00533 2/20 0.40
CDK8 P49336 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9517068 0.92 CASP3 (0.47) CASP3P4HTMSMN1; SMN2PTGS2HTT
SCHEMBL9516171 0.88 SMN1; SMN2 (0.46) CASP3P4HTMSMN1; SMN2MEN1KMT2A
SCHEMBL9519106 0.88 EGFR (0.50) P4HTMPTGS2PTGS1EGFR
SCHEMBL9519516 0.86 HTT (0.60) CASP3P4HTMHTT
SCHEMBL27379257 0.85 P4HTM (0.50) CASP3P4HTMPTGS2PTGS1EGFR
SCHEMBL8869795 0.84 P4HTM (0.51) CASP3P4HTMSMN1; SMN2HTTNAMPT
SCHEMBL9140003 0.83 P4HTM (0.52) CASP3P4HTMSMN1; SMN2PTGS2HTT
SCHEMBL9517927 0.82 P4HTM (0.42) CASP3P4HTMPTGS2
SCHEMBL9018408 0.81 SMN1; SMN2 (0.46) CASP3P4HTMSMN1; SMN2PTGS2HTT
SCHEMBL9139358 0.81 P4HTM (0.50) CASP3P4HTMSMN1; SMN2PTGS2HTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0567997-A1 4- or 5-(sulf)imido- and (sulfon)amidopyridines and their pyridine-N-oxides, process for their preparation and their use as pharmaceutical HOECHST AKTIENGESELLSCHAFT (DE) 1993-11-03 EP disclosed