SCHEMBL9520385

SCHEMBL9520385

Cc1oc(-c2ccccc2)nc1CCC(=O)c1ccc(/C=C2/SC(=O)NC2=O)nc1

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
PPARG P37231 16/20 0.41
PPARA Q07869 16/20 0.41
KDM4E B2RXH2 1/20 0.41
KCNH2 Q12809 1/20 0.41
FFAR1 O14842 1/20 0.40
PIK3CG P48736 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9520389 1.00 PPARG (0.41) PPARGPPARAKDM4EKCNH2FFAR1
SCHEMBL9520097 0.90 KDM4E (0.45) PPARGPPARAKDM4EKCNH2PIK3CG
SCHEMBL9520104 0.90 KDM4E (0.45) PPARGPPARAKDM4EKCNH2PIK3CG
SCHEMBL9521137 0.83 PIM1 (0.49) PPARGPPARAKDM4E
SCHEMBL9521141 0.83 PIM1 (0.49) PPARGPPARAKDM4E
SCHEMBL9523273 0.82 KDM4E (0.50) PPARGPPARAKDM4EFFAR1
SCHEMBL9379554 0.81 HPGD (0.54) KDM4E
SCHEMBL9379550 0.81 HPGD (0.54) KDM4E
SCHEMBL9521885 0.81 PTPN1 (0.43) PPARGPPARA
SCHEMBL9521889 0.81 PTPN1 (0.43) PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0332332-B1 HYPOGLYCEMIC THIAZOLIDINEDIONE DERIVATIVES PFIZER INC. (US) 1993-03-31 EP disclosed
WO-1989008651-A1 HYPOGLYCEMIC THIAZOLIDINEDIONE DERIVATIVES PFIZER INC. (US) 1989-09-21 WO disclosed