SCHEMBL9520686

SCHEMBL9520686

Cc1oc(-c2ccccc2)nc1CCC(O[Si](C)(C)C(C)(C)C)c1ccc(Br)s1

nearest known ligand 0.44

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PPARG P37231 17/20 0.44
PPARA Q07869 17/20 0.44
PPARD Q03181 6/20 0.44
HRH3 Q9Y5N1 1/20 0.40
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9721238 0.92 PPARA (0.38) PPARGPPARAPPARDKDM4E
SCHEMBL9521721 0.86 PPARG (0.44) PPARGPPARAPPARDHRH3KDM4E
SCHEMBL9520406 0.80 KDM4E (0.47) PPARGPPARAPPARDHRH3KDM4E
SCHEMBL9008053 0.79 PPARA (0.47) PPARGPPARAPPARDHRH3KDM4E
SCHEMBL9520129 0.79 PPARG (0.40) PPARGPPARAPPARD
SCHEMBL9521119 0.78 PPARG (0.38) PPARGPPARAPPARDHRH3
SCHEMBL9521124 0.78 PPARG (0.38) PPARGPPARAPPARDHRH3
SCHEMBL9721263 0.78 MAPT (0.36) PPARGPPARAPPARDKDM4E
SCHEMBL7879102 0.77 PPARG (0.46) PPARGPPARAPPARDHRH3KDM4E
SCHEMBL7879105 0.77 PPARG (0.46) PPARGPPARAPPARDHRH3KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0332332-B1 HYPOGLYCEMIC THIAZOLIDINEDIONE DERIVATIVES PFIZER INC. (US) 1993-03-31 EP disclosed
US-5130379-A Anticholesterol agents and antidiabetic agents PFIZER INC. (US) 1992-07-14 US disclosed
US-5036079-A Anticholesterol PFIZER INC. (US) 1991-07-30 US disclosed
WO-1991003474-A1 HYPOGLYCEMIC THIAZOLIDINEDIONE DERIVATIVES PFIZER INC. (US) 1991-03-21 WO disclosed
WO-1989008651-A1 HYPOGLYCEMIC THIAZOLIDINEDIONE DERIVATIVES PFIZER INC. (US) 1989-09-21 WO disclosed
EP-0332332-A1 Hypoglycemic thiazolidinedione derivatives PFIZER INC. (US) 1989-09-13 EP disclosed