SCHEMBL9520129

SCHEMBL9520129

Cc1oc(-c2ccccc2)nc1CCC(O[Si](C)(C)C(C)(C)C)c1ccc(CC2SC(=O)NC2=O)s1

nearest known ligand 0.40

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PPARG P37231 18/20 0.40
PPARA Q07869 17/20 0.40
PPARD Q03181 6/20 0.40
LIPG Q9Y5X9 1/20 0.37
FFAR1 O14842 1/20 0.37
CYP2C9 P11712 2/20 0.37
CYP3A4 P08684 1/20 0.37
KCNH2 Q12809 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9721194 0.94 PPARA (0.37) PPARGPPARAPPARDLIPGFFAR1
SCHEMBL9878676 0.81 PPARA (0.36) PPARGPPARAPPARDFFAR1
SCHEMBL9520686 0.79 PPARG (0.44) PPARGPPARAPPARD
SCHEMBL9521721 0.78 PPARG (0.44) PPARGPPARAPPARD
SCHEMBL9520439 0.78 PPARG (0.43) PPARGPPARAPPARDFFAR1CYP2C9
SCHEMBL9521124 0.78 PPARG (0.38) PPARGPPARAPPARDKCNH2
SCHEMBL9521119 0.78 PPARG (0.38) PPARGPPARAPPARDKCNH2
SCHEMBL7871522 0.77 PPARG (0.46) PPARGPPARAPPARDFFAR1CYP2C9
SCHEMBL7871527 0.77 PPARG (0.46) PPARGPPARAPPARDFFAR1CYP2C9
SCHEMBL7722467 0.75 PPARG (0.42) PPARGPPARAPPARD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0332332-B1 HYPOGLYCEMIC THIAZOLIDINEDIONE DERIVATIVES PFIZER INC. (US) 1993-03-31 EP disclosed
US-5130379-A Anticholesterol agents and antidiabetic agents PFIZER INC. (US) 1992-07-14 US disclosed
US-5036079-A Anticholesterol PFIZER INC. (US) 1991-07-30 US disclosed
WO-1991003474-A1 HYPOGLYCEMIC THIAZOLIDINEDIONE DERIVATIVES PFIZER INC. (US) 1991-03-21 WO disclosed
EP-0332332-A1 Hypoglycemic thiazolidinedione derivatives PFIZER INC. (US) 1989-09-13 EP disclosed