SCHEMBL9520918

SCHEMBL9520918

O=CC=C(c1ccc(Cl)cc1)c1ccc(Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 3/20 0.48
CES1 P23141 3/20 0.48
TSHR P16473 2/20 0.46
ALOX15 P16050 1/20 0.46
CA1 P00915 2/20 0.44
CA2 P00918 2/20 0.44
HSD17B10 Q99714 1/20 0.42
PTGS2 P35354 1/20 0.42
MAPK1 P28482 2/20 0.41
GSK3B P49841 2/20 0.41
SRD5A2 P31213 1/20 0.41
BCL2L1 Q07817 1/20 0.41
L3MBTL1 Q9Y468 2/20 0.41
CYP3A4 P08684 1/20 0.41
ATM Q13315 1/20 0.41
LMNA P02545 3/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
KDM4E B2RXH2 1/20 0.40
CYP1A2 P05177 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10579805 0.92 CES2 (0.55) CES2CES1TSHRALOX15PTGS2
SCHEMBL29016164 0.92 CES2 (0.55) CES2CES1TSHRALOX15PTGS2
SCHEMBL25321662 0.85 ALDH1A1 (0.56) TSHRALOX15HSD17B10MAPK1BCL2L1
SCHEMBL9421060 0.85 CES2 (0.43) CES2CES1TSHRALOX15CA1
SCHEMBL9421070 0.85 CES2 (0.43) CES2CES1TSHRALOX15CA1
SCHEMBL11137766 0.81 MAPT (0.51) TSHRALOX15PTGS2L3MBTL1LMNA
SCHEMBL12676349 0.81 BCL2L1 (0.34) CES2CES1TSHRALOX15CA1
SCHEMBL11137762 0.81 MAPT (0.51) TSHRALOX15PTGS2L3MBTL1LMNA
SCHEMBL5077542 0.80 ABCG2 (0.55) TSHRCA1CA2CYP3A4LMNA
SCHEMBL2559260 0.79 CES2 (0.46) CES2CES1TSHRALOX15CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104926629-B Domino reaction is utilized to prepare the green method of 3,3-diaryl acrylic aldehyde 江苏科本医药化学有限公司 2016-06-22 CN claimed
CN-104926629-A Environment-friendly method for preparing 3,3-diaryl acrolein by utilizing domino reaction JIANGSU COBEN PHARMACEUTICAL CO LTD 2015-09-23 CN claimed
CN-104926629-B Domino reaction is utilized to prepare the green method of 3,3-diaryl acrylic aldehyde 江苏科本医药化学有限公司 2016-06-22 CN disclosed
CN-104926629-A Environment-friendly method for preparing 3,3-diaryl acrolein by utilizing domino reaction JIANGSU COBEN PHARMACEUTICAL CO LTD 2015-09-23 CN disclosed
EP-0299379-B1 PENTADIENAMIDE PAF-ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
US-4975438-A ANTICOAGULANT HOFFMANN-LA ROCHE INC. (US) 1990-12-04 US disclosed
EP-0299379-A1 Pentadienamide PAF-antagonists F. HOFFMANN-LA ROCHE AG (CH) 1989-01-18 EP disclosed
US-4788206-A CARDIOVASCULAR DISORDERS, PLATELETS HOFFMANN-LA ROCHE INC. (US) 1988-11-29 US disclosed