SCHEMBL9521022

SCHEMBL9521022

COc1cccc(/C(=C/C=O)c2cccc(F)c2)c1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.61
RAB9A P51151 3/20 0.61
ALDH1A1 P00352 3/20 0.57
CES2 O00748 1/20 0.50
CES1 P23141 1/20 0.50
KDM4E B2RXH2 2/20 0.49
NFE2L2 Q16236 1/20 0.49
SMN1; SMN2 Q16637 1/20 0.48
PDE4A P27815 1/20 0.48
PDE4B Q07343 1/20 0.48
PDE4C Q08493 1/20 0.48
PDE4D Q08499 1/20 0.48
PARP1 P09874 1/20 0.47
PTAFR P25105 2/20 0.47
MTNR1A P48039 3/20 0.47
MTNR1B P49286 3/20 0.47
TSHR P16473 1/20 0.47
NPSR1 Q6W5P4 1/20 0.47
POLB P06746 1/20 0.46
ABCG2 Q9UNQ0 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9521029 1.00 NPC1 (0.61) NPC1RAB9AALDH1A1CES2CES1
SCHEMBL10399040 1.00 NPC1 (0.61) NPC1RAB9AALDH1A1CES2CES1
SCHEMBL9519728 0.91 CES2 (0.59) NPC1RAB9ACES2CES1SMN1; SMN2
SCHEMBL9521397 0.90 NPC1 (0.49) NPC1RAB9AALDH1A1CES2CES1
SCHEMBL9521399 0.90 NPC1 (0.49) NPC1RAB9AALDH1A1CES2CES1
SCHEMBL9520429 0.86 MTNR1A (0.57) NPC1RAB9AALDH1A1CES2CES1
SCHEMBL9520444 0.86 MTNR1A (0.57) NPC1RAB9AALDH1A1CES2CES1
SCHEMBL9520437 0.86 MTNR1A (0.57) NPC1RAB9AALDH1A1CES2CES1
SCHEMBL9520017 0.86 CES2 (0.55) NPC1RAB9ACES2CES1KDM4E
SCHEMBL10521631 0.84 NPC1 (0.56) NPC1RAB9AALDH1A1CES2CES1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0299379-B1 PENTADIENAMIDE PAF-ANTAGONISTS F. HOFFMANN-LA ROCHE AG (CH) 1993-04-21 EP disclosed
US-4975438-A ANTICOAGULANT HOFFMANN-LA ROCHE INC. (US) 1990-12-04 US disclosed
EP-0299379-A1 Pentadienamide PAF-antagonists F. HOFFMANN-LA ROCHE AG (CH) 1989-01-18 EP disclosed
US-4788206-A CARDIOVASCULAR DISORDERS, PLATELETS HOFFMANN-LA ROCHE INC. (US) 1988-11-29 US disclosed