SCHEMBL9522296

SCHEMBL9522296

N#CC(C(=O)Nc1ccccc1)C(=O)c1nn(-c2ccccc2)c2c1CSc1ccc(C(=O)NCC(=O)O)cc1-2

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
TP53 P04637 7/20 0.37
MAPT P10636 6/20 0.37
LMNA P02545 2/20 0.37
PTPRC P08575 2/20 0.36
CTSL P07711 1/20 0.36
PTPN13 Q12923 1/20 0.36
ALDH1A1 P00352 2/20 0.33
TSHR P16473 1/20 0.32
NPSR1 Q6W5P4 1/20 0.32
HSD17B10 Q99714 1/20 0.32
DGAT1 O75907 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9523089 0.93 TP53 (0.38) TP53MAPTLMNAALDH1A1
SCHEMBL9523890 0.91 TP53 (0.35) TP53MAPTLMNAALDH1A1TSHR
SCHEMBL9522751 0.89 TP53 (0.38) TP53MAPTLMNAALDH1A1
SCHEMBL9523673 0.88 TP53 (0.35) TP53MAPTLMNADGAT1
SCHEMBL9522441 0.88 TP53 (0.44) TP53MAPTLMNAALDH1A1NPSR1
SCHEMBL9176686 0.87 PTPRC (0.37) LMNAPTPRCCTSLPTPN13ALDH1A1
SCHEMBL9522233 0.87 KMT2A (0.44) TP53MAPTLMNAALDH1A1NPSR1
SCHEMBL9525929 0.86 DGAT1 (0.37) TP53MAPTLMNACTSLDGAT1
SCHEMBL9523140 0.86 TP53 (0.37) TP53MAPTLMNAALDH1A1NPSR1
SCHEMBL9523576 0.86 TP53 (0.34) TP53MAPTLMNAALDH1A1TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0420883-B1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION ERBA CARLO SPA (IT) 1993-11-03 EP disclosed
US-5166152-A Immunostimulants, bactericides, viricides, antitumor agents FARMITALIA CARLO ERBA S.R.L. (IT) 1992-11-24 US disclosed
EP-0420883-A1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION. ERBA CARLO SPA (IT) 1991-04-10 EP disclosed
WO-1989012638-A1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1989-12-28 WO disclosed