SCHEMBL9525929

SCHEMBL9525929

CC(C)C[C@H](NC(=O)c1ccc2c(c1)-c1c(c(C(=O)C(C#N)C(=O)Nc3ccccc3)nn1-c1ccccc1)CS2)C(=O)O

nearest known ligand 0.37

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 1/20 0.37
F3 P13726 3/20 0.37
CTSL P07711 9/20 0.36
CTSB P07858 4/20 0.36
CTSS P25774 3/20 0.36
CTSK P43235 3/20 0.36
GRN P28799 1/20 0.35
SORT1 Q99523 1/20 0.35
MAPK14 Q16539 1/20 0.35
TP53 P04637 2/20 0.34
MAPT P10636 2/20 0.34
LMNA P02545 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9523565 0.94 TAS1R3 (0.36) CTSLCTSBCTSSCTSKMAPK14
SCHEMBL9523673 0.91 TP53 (0.35) DGAT1MAPK14TP53MAPTLMNA
SCHEMBL9174778 0.88 MAPK14 (0.40) DGAT1F3CTSLCTSBCTSS
SCHEMBL9523140 0.88 TP53 (0.37) MAPK14TP53MAPTLMNA
SCHEMBL9522296 0.86 TP53 (0.37) DGAT1CTSLTP53MAPTLMNA
SCHEMBL9523890 0.86 TP53 (0.35) TP53MAPTLMNA
SCHEMBL9523403 0.86 F3 (0.36) DGAT1F3CTSLGRNSORT1
SCHEMBL9523089 0.85 TP53 (0.38) TP53MAPTLMNA
SCHEMBL9522233 0.85 KMT2A (0.44) TP53MAPTLMNA
SCHEMBL9522441 0.85 TP53 (0.44) TP53MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0420883-B1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION ERBA CARLO SPA (IT) 1993-11-03 EP disclosed
US-5166152-A Immunostimulants, bactericides, viricides, antitumor agents FARMITALIA CARLO ERBA S.R.L. (IT) 1992-11-24 US disclosed
EP-0420883-A1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION. ERBA CARLO SPA (IT) 1991-04-10 EP disclosed
WO-1989012638-A1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1989-12-28 WO disclosed