SCHEMBL9522966

SCHEMBL9522966

N#CC(C(=O)Nc1ccccc1)C(=O)c1nn(-c2ccccc2)c2c1CSc1ccc(NC(=O)CN)cc1-2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TP53 P04637 6/20 0.34
MAPT P10636 3/20 0.34
LMNA P02545 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
ALDH1A1 P00352 2/20 0.34
NPSR1 Q6W5P4 2/20 0.34
PIK3CD O00329 2/20 0.34
PIK3R2 O00459 2/20 0.34
PIK3CA P42336 2/20 0.34
PIK3CB P42338 2/20 0.34
PIK3CG P48736 2/20 0.34
PIK3R5 Q8WYR1 2/20 0.34
PIK3R3 Q92569 2/20 0.34
TSHR P16473 1/20 0.34
HSD17B10 Q99714 1/20 0.34
IKBKB O14920 3/20 0.33
TERT O14746 1/20 0.33
CARM1 Q86X55 1/20 0.33
KLKB1 P03952 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9523576 0.93 TP53 (0.34) TP53MAPTLMNACA1CA2
SCHEMBL9524294 0.92 ADORA3 (0.34) TP53MAPTLMNAALDH1A1NPSR1
SCHEMBL9523480 0.88 MAPT (0.34) TP53MAPTLMNACA1CA2
SCHEMBL9316111 0.88 PIK3CD (0.38) TP53MAPTLMNACA1CA2
SCHEMBL9316496 0.88 MEN1 (0.40) TP53MAPTLMNAALDH1A1
SCHEMBL9316080 0.88 TP53 (0.37) TP53MAPTLMNACA1CA2
SCHEMBL9522373 0.86 AURKB (0.34) TP53MAPTLMNAPIK3CDPIK3R2
SCHEMBL9316680 0.86 MAPT (0.45) TP53MAPTLMNAALDH1A1PIK3CD
SCHEMBL9523890 0.86 TP53 (0.35) TP53MAPTLMNACA1CA2
SCHEMBL9831280 0.86 PIK3CD (0.37) TP53MAPTLMNAALDH1A1NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0420883-B1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION ERBA CARLO SPA (IT) 1993-11-03 EP disclosed
US-5166152-A Immunostimulants, bactericides, viricides, antitumor agents FARMITALIA CARLO ERBA S.R.L. (IT) 1992-11-24 US disclosed