SCHEMBL9524294

SCHEMBL9524294

N#CC(C(=O)Nc1ccccc1)C(=O)c1nn(-c2ccccc2)c2c1CSc1ccc(NC(=O)CCC(=O)O)cc1-2

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADORA3 P0DMS8 1/20 0.34
ADORA2A P29274 1/20 0.34
ADORA1 P30542 1/20 0.34
TP53 P04637 5/20 0.34
MAPT P10636 4/20 0.34
LMNA P02545 1/20 0.34
MEN1 O00255 4/20 0.33
KMT2A Q03164 4/20 0.33
POLB P06746 3/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
CYP1A2 P05177 1/20 0.33
PIK3CD O00329 1/20 0.33
PIK3R2 O00459 1/20 0.33
PIK3CA P42336 1/20 0.33
PIK3CB P42338 1/20 0.33
PIK3CG P48736 1/20 0.33
PIK3R5 Q8WYR1 1/20 0.33
PIK3R3 Q92569 1/20 0.33
ALDH1A1 P00352 4/20 0.33
KDM4E B2RXH2 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9523576 0.94 TP53 (0.34) TP53MAPTLMNAMEN1KMT2A
SCHEMBL9522966 0.92 TP53 (0.34) TP53MAPTLMNAPIK3CDPIK3R2
SCHEMBL9523480 0.88 MAPT (0.34) TP53MAPTLMNAPIK3CDPIK3R2
SCHEMBL9837477 0.88 POLB (0.39) ADORA3ADORA2AADORA1TP53MAPT
SCHEMBL9316496 0.87 MEN1 (0.40) TP53MAPTLMNAMEN1KMT2A
SCHEMBL9316080 0.87 TP53 (0.37) TP53MAPTLMNAPIK3CDPIK3R2
SCHEMBL9523670 0.86 MAPT (0.33) TP53MAPTLMNAMEN1KMT2A
SCHEMBL9522373 0.86 AURKB (0.34) TP53MAPTLMNAPIK3CDPIK3R2
SCHEMBL9316111 0.86 PIK3CD (0.38) TP53MAPTLMNAPIK3CDPIK3R2
SCHEMBL9523890 0.86 TP53 (0.35) TP53MAPTLMNAMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0420883-B1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION ERBA CARLO SPA (IT) 1993-11-03 EP disclosed
US-5166152-A Immunostimulants, bactericides, viricides, antitumor agents FARMITALIA CARLO ERBA S.R.L. (IT) 1992-11-24 US disclosed
EP-0420883-A1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION. ERBA CARLO SPA (IT) 1991-04-10 EP disclosed
WO-1989012638-A1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION FARMITALIA CARLO ERBA S.R.L. (IT) 1989-12-28 WO disclosed