SCHEMBL9523726

SCHEMBL9523726

CCOC(=O)C(=O)Nc1ccc2c(c1)-c1c(c(C(=O)C(C#N)C(=O)Nc3cccc([N+](=O)[O-])c3)nn1-c1ccccc1)CS2

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 1/20 0.39
CA2 P00918 1/20 0.39
ALDH1A1 P00352 4/20 0.37
KMT2A Q03164 8/20 0.37
MEN1 O00255 6/20 0.37
NPC1 O15118 2/20 0.37
RAB9A P51151 1/20 0.37
ALOX12 P18054 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4D Q08499 1/20 0.35
HSP90AA1 P07900 1/20 0.34
PKM P14618 1/20 0.34
HPGD P15428 1/20 0.34
CCR6 P51684 1/20 0.34
NPSR1 Q6W5P4 1/20 0.34
APOBEC3G Q9HC16 1/20 0.34
KDM4E B2RXH2 2/20 0.34
LMNA P02545 2/20 0.34
MAPT P10636 2/20 0.34
MAPK1 P28482 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9523720 0.92 MEN1 (0.37) CA1CA2ALDH1A1KMT2AMEN1
SCHEMBL9316085 0.92 MAPT (0.37) CA1CA2ALDH1A1KMT2AKDM4E
SCHEMBL9522378 0.90 RIPK1 (0.38) ALDH1A1KMT2AMEN1LMNAMAPT
SCHEMBL9525898 0.89 MAPT (0.40) ALDH1A1KMT2AHPGDNPSR1KDM4E
SCHEMBL9522532 0.88 MAPT (0.39) ALDH1A1HPGDNPSR1KDM4ELMNA
SCHEMBL9525574 0.88 LMNA (0.37) ALDH1A1KMT2AMEN1LMNAMAPT
SCHEMBL9316548 0.87 MEN1 (0.40) ALDH1A1KMT2AMEN1NPC1RAB9A
SCHEMBL9316080 0.85 TP53 (0.37) CA1CA2LMNAMAPTTP53
SCHEMBL9834297 0.83 MAPK14 (0.40) CA1CA2ALDH1A1KMT2AMEN1
SCHEMBL9522374 0.82 RIPK1 (0.39) ALDH1A1KMT2AMEN1KDM4ELMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0420883-B1 TRICYCLIC 3-OXO-PROPANENITRILE DERIVATIVES AND PROCESS FOR THEIR PREPARATION ERBA CARLO SPA (IT) 1993-11-03 EP disclosed
US-5166152-A Immunostimulants, bactericides, viricides, antitumor agents FARMITALIA CARLO ERBA S.R.L. (IT) 1992-11-24 US disclosed