SCHEMBL9523866

SCHEMBL9523866

CCCCn1nnc2cc(C=O)ccc21

nearest known ligand 0.61

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
HCAR3 P49019 7/20 0.61
SLC9A1 P19634 7/20 0.57
GRM2 Q14416 1/20 0.43
CYP2A6 P11509 2/20 0.39
PTGER4 P35408 1/20 0.37
ALDH1A1 P00352 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14931778 0.86 HCAR3 (0.48) HCAR3SLC9A1CYP2A6
SCHEMBL19088929 0.86 HCAR3 (0.45) HCAR3SLC9A1CYP2A6
SCHEMBL14931736 0.86 HCAR3 (0.45) HCAR3SLC9A1CYP2A6
SCHEMBL28473872 0.84 HCAR3 (0.49) HCAR3SLC9A1CYP2A6
SCHEMBL28468120 0.82 HCAR3 (0.46) HCAR3SLC9A1CYP2A6
SCHEMBL14942089 0.81 HCAR3 (0.42) HCAR3SLC9A1CYP2A6PTGER4
SCHEMBL28470307 0.80 HCAR3 (0.45) HCAR3SLC9A1
SCHEMBL15823043 0.80 HCAR3 (0.41) HCAR3SLC9A1CYP2A6
SCHEMBL28465267 0.80 HCAR3 (0.46) HCAR3SLC9A1CYP2A6PTGER4ALDH1A1
SCHEMBL19848522 0.79 SLC9A1 (0.64) HCAR3SLC9A1GRM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1022184-C Process for preparing (1 H-imidzol-1-ylmethyl) substituted benzotriazole derivatives JANSSEN PHARMACEUTICA NV (BE) 1993-09-22 CN disclosed
EP-0293978-B1 (1H-AZOL-1-YLMETHYL)SUBSTITUTED BENZOTRIAZOLE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1993-09-15 EP disclosed
US-5039677-A Estrogen inhibitor JANSSEN PHARMACEUTICA N.V. (CA) 1991-08-13 US disclosed
US-4943574-A AROMATASE INHIBITORS, ESTROGEN DISORDERS JANSSEN PHARMACEUTICA N.V. (BE) 1990-07-24 US disclosed
CN-88103408-A Process for preparing (1H-oxazol-1-ylmethyl) substituted benzotriazole derivatives 1988-12-14 CN disclosed
EP-0293978-A2 (1H-azol-1-ylmethyl)substituted benzotriazole derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1988-12-07 EP disclosed