SCHEMBL9523911

SCHEMBL9523911

Cc1cccc(C2CC(C)(C)Oc3ccc(C#N)cc32)[n+]1[O-]

nearest known ligand 0.38

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
SIRT2 Q8IXJ6 4/20 0.38
ABCB1 P08183 8/20 0.38
SIRT1 Q96EB6 2/20 0.36
KDM4E B2RXH2 1/20 0.36
ABCC9 O60706 5/20 0.35
ABCC8 Q09428 2/20 0.35
KCNJ11 Q14654 2/20 0.35
KCNJ8 Q15842 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP2D6 P10635 1/20 0.35
CYP2C9 P11712 1/20 0.35
CYP2C19 P33261 1/20 0.35
LMNA P02545 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525708 0.88 ABCC9 (0.39) SIRT2ABCB1SIRT1ABCC9
SCHEMBL9525278 0.88 SIRT2 (0.38) SIRT2ABCB1SIRT1KDM4EABCC9
SCHEMBL8174728 0.83 ABCB1 (0.40) SIRT2ABCB1KDM4EABCC9ABCC8
SCHEMBL8174878 0.83 ABCB1 (0.40) SIRT2ABCB1KDM4EABCC9ABCC8
SCHEMBL8174399 0.83 ABCB1 (0.40) SIRT2ABCB1KDM4EABCC9ABCC8
SCHEMBL9524832 0.83 ABCB1 (0.37) SIRT2ABCB1KDM4EABCC9ABCC8
SCHEMBL9525021 0.83 ABCB1 (0.40) ABCB1KDM4EABCC9ABCC8KCNJ11
SCHEMBL9523798 0.81 ABCB1 (0.40) SIRT2ABCB1KDM4EABCC9ABCC8
SCHEMBL9525704 0.80 ABCB1 (0.39) SIRT2ABCB1KDM4EABCC9ABCC8
SCHEMBL9525130 0.80 ABCC9 (0.40) ABCB1ABCC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0298452-B1 2H-1-BENZOPYRANE DERIVATIVES SUBSTITUTED IN POSITION 4 BY ARYL OR N-HETEROARYL F. HOFFMANN-LA ROCHE AG (CH) 1993-06-30 EP claimed
US-5118694-A Hypotensive agents; treatment for cardiovascular and muscular disorders HOFFMANN-LA ROCHE INC. (US) 1992-06-02 US disclosed
US-4971982-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, SMOOTH MUSCLE DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-11-20 US disclosed