SCHEMBL9524111

SCHEMBL9524111

COc1cc(/C=C/C(=O)Oc2ccc([N+](=O)[O-])cc2)cc(OC)c1OC

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KRAS P01116 3/20 0.72
HTR1A P08908 2/20 0.68
PTGS2 P35354 2/20 0.67
ALDH1A1 P00352 3/20 0.61
HTT P42858 3/20 0.61
MAPT P10636 3/20 0.61
LMNA P02545 2/20 0.61
TUBB4A P04350 2/20 0.55
TUBB P07437 2/20 0.55
TUBA3C P0DPH7 2/20 0.55
TUBA1B P68363 2/20 0.55
TUBA4A P68366 2/20 0.55
TUBB4B P68371 2/20 0.55
TUBB3 Q13509 2/20 0.55
TUBB2A Q13885 2/20 0.55
TUBB8 Q3ZCM7 2/20 0.55
TUBA3E Q6PEY2 2/20 0.55
TUBA1A Q71U36 2/20 0.55
TUBA1C Q9BQE3 2/20 0.55
TUBB6 Q9BUF5 2/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524117 1.00 KRAS (0.72) KRASHTR1APTGS2ALDH1A1HTT
SCHEMBL760063 0.90 KRAS (0.72) KRASHTR1APTGS2ALDH1A1HTT
SCHEMBL9523755 0.88 PTGS2 (0.69) KRASPTGS2ALDH1A1MAPTGAA
SCHEMBL9523759 0.88 PTGS2 (0.69) KRASPTGS2ALDH1A1MAPTGAA
SCHEMBL1597196 0.85 MAPT (0.66) PTGS2ALDH1A1HTTMAPTLMNA
SCHEMBL30839393 0.85 MAPT (0.66) PTGS2ALDH1A1HTTMAPTLMNA
SCHEMBL9522624 0.83 CYP19A1 (0.55) KRASPTGS2ALDH1A1HTTMAPT
SCHEMBL9522627 0.83 CYP19A1 (0.55) KRASPTGS2ALDH1A1HTTMAPT
SCHEMBL9478353 0.83 MAOB (0.73) KRASPTGS2ALDH1A1MAPTLMNA
SCHEMBL9478343 0.83 MAOB (0.73) KRASPTGS2ALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0354583-B1 DC-88A derivatives KYOWA HAKKO KOGYO KK (JP) 1993-11-03 EP disclosed
US-5117006-A DC-88A DERIVATIVES USEFUL AS ANTITUMOR AGENTS KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-05-26 US disclosed
US-5084468-A Antitumor agents KYOWA HAKKO KOGYO CO., LTD. (JP) 1992-01-28 US disclosed
EP-0354583-A1 DC-88A derivatives KYOWA HAKKO KOGYO CO., LTD. (JP) 1990-02-14 EP disclosed