SCHEMBL9525469

SCHEMBL9525469

COC(=O)CC[C@H](NC(=O)c1cccc(CCC2CNc3nc(NC(=O)C(C)(C)C)nc(O)c3C2)c1)C(=O)OC

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
GART P22102 4/20 0.41
DHFR P00374 3/20 0.36
KDR P35968 2/20 0.34
ROCK2 O75116 1/20 0.33
FNTA P49354 3/20 0.32
FNTB P49356 3/20 0.32
MAPK14 Q16539 1/20 0.32
BCHE P06276 1/20 0.32
ACHE P22303 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10568483 1.00 GART (0.41) GARTDHFRKDRROCK2FNTA
SCHEMBL8819377 0.91 GART (0.39) GARTDHFRROCK2
SCHEMBL8819374 0.91 GART (0.39) GARTDHFRROCK2
SCHEMBL9524143 0.88 GART (0.38) GARTDHFR
SCHEMBL9524154 0.88 GART (0.38) GARTDHFR
SCHEMBL8819372 0.87 GART (0.40) GARTDHFRKDRROCK2MAPK14
SCHEMBL8819376 0.87 GART (0.40) GARTDHFRKDRROCK2MAPK14
SCHEMBL9381356 0.86 GART (0.36) GARTDHFR
SCHEMBL9381360 0.86 GART (0.36) GARTDHFR
SCHEMBL9383820 0.86 DHFR (0.46) GARTDHFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0327190-B1 Pyrido(2,3-d)pyrimidine derivatives UNIV PRINCETON (US) 1993-12-08 EP disclosed
US-4889859-A ANTITUMOR AGENTS THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-12-26 US disclosed
EP-0327190-A1 Pyrido(2,3-d)pyrimidine derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-08-09 EP disclosed