SCHEMBL9524342

SCHEMBL9524342

COc1ccc(COC(=O)Sc2cc(C)cc(C)n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.43
CYP1A2 P05177 1/20 0.43
CYP3A4 P08684 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
POLB P06746 4/20 0.41
LMNA P02545 2/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
ALDH1A1 P00352 4/20 0.41
MAOB P27338 1/20 0.40
MMP13 P45452 1/20 0.40
DHODH Q02127 2/20 0.40
TSPO P30536 1/20 0.40
KDM4E B2RXH2 3/20 0.39
MAPT P10636 3/20 0.39
HPGD P15428 2/20 0.39
HSD17B10 Q99714 2/20 0.39
GAA P10253 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
PHGDH O43175 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5521119 0.83 MAOB (0.45) HTTPOLBLMNASMN1; SMN2ALDH1A1
SCHEMBL29009279 0.70 ALDH1A1 (0.53) HTTPOLBSMN1; SMN2ALDH1A1KDM4E
SCHEMBL11853555 0.69 ALDH1A1 (0.40) HTTPOLBLMNASMN1; SMN2ALDH1A1
SCHEMBL8713714 0.68 NPSR1 (0.36) CYP1A2CYP3A4CYP2C9CYP2C19SMN1; SMN2
SCHEMBL7268455 0.68 HPGD (0.48) HTTSMN1; SMN2ALDH1A1KDM4EMAPT
SCHEMBL3758807 0.68 ALDH1A1 (0.60) HTTPOLBSMN1; SMN2ALDH1A1MAPT
SCHEMBL292834 0.68 ALDH1A1 (0.60) HTTPOLBSMN1; SMN2ALDH1A1MAPT
SCHEMBL19514751 0.67 POLB (0.49) HTTPOLBSMN1; SMN2ALDH1A1KDM4E
SCHEMBL4710453 0.67 SMN1; SMN2 (0.69) HTTCYP1A2CYP3A4LMNASMN1; SMN2
SCHEMBL6403295 0.66 ALDH1A1 (0.58) HTTPOLBSMN1; SMN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0249170-B1 CEPHEM COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-17 EP disclosed
US-4921851-A Cephem compounds, their production and use TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1990-05-01 US disclosed
EP-0249170-A2 Cephem compounds, their production and use Takeda Chemical Industries, Ltd. (JP) 1987-12-16 EP disclosed
US-4546176-A 7-Carboxymethoxyphenylacetamido-3-cephem derivatives and antibacterial preparations containing the same EISAI CO., LTD. (JP) 1985-10-08 US disclosed