SCHEMBL9524433

SCHEMBL9524433

O=[N+]([O-])c1cc(C(Br)c2ccccc2)ccc1Cl

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
VCAM1 P19320 8/20 0.50
MEN1 O00255 4/20 0.50
KMT2A Q03164 4/20 0.50
MAPT P10636 2/20 0.50
HTT P42858 2/20 0.50
CYP1A2 P05177 1/20 0.50
CYP3A4 P08684 1/20 0.50
CYP2D6 P10635 1/20 0.50
CYP2C9 P11712 1/20 0.50
CYP2C19 P33261 1/20 0.50
RECQL P46063 1/20 0.50
LMNA P02545 3/20 0.47
GAA P10253 1/20 0.47
SMN1; SMN2 Q16637 4/20 0.46
NPSR1 Q6W5P4 2/20 0.46
ALDH1A1 P00352 3/20 0.44
SLC25A1 P53007 1/20 0.43
GRM8 O00222 1/20 0.43
GRM6 O15303 1/20 0.43
GRM4 Q14833 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9523568 0.81 VCAM1 (0.54) VCAM1MEN1KMT2AMAPTHTT
SCHEMBL31067431 0.81 VCAM1 (0.54) VCAM1MEN1KMT2AMAPTHTT
SCHEMBL11712759 0.79 VCAM1 (0.51) VCAM1MEN1KMT2AMAPTHTT
SCHEMBL2998296 0.76 VCAM1 (0.54) VCAM1MEN1KMT2AMAPTHTT
SCHEMBL22440060 0.76 VCAM1 (0.54) VCAM1MEN1KMT2AMAPTHTT
SCHEMBL14092697 0.76 TSHR (0.61) VCAM1MAPTHTTCYP1A2CYP3A4
SCHEMBL15791936 0.75 VCAM1 (0.45) VCAM1MEN1KMT2AMAPTHTT
SCHEMBL6745454 0.75 VCAM1 (0.49) VCAM1MEN1KMT2AMAPTHTT
SCHEMBL16952092 0.75 VCAM1 (0.49) VCAM1MEN1KMT2AMAPTHTT
SCHEMBL28044205 0.75 HPGD (0.44) VCAM1MEN1KMT2AMAPTCYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0293978-B1 (1H-AZOL-1-YLMETHYL)SUBSTITUTED BENZOTRIAZOLE DERIVATIVES JANSSEN PHARMACEUTICA N.V. (BE) 1993-09-15 EP disclosed
US-5039677-A Estrogen inhibitor JANSSEN PHARMACEUTICA N.V. (CA) 1991-08-13 US disclosed
US-4943574-A AROMATASE INHIBITORS, ESTROGEN DISORDERS JANSSEN PHARMACEUTICA N.V. (BE) 1990-07-24 US disclosed
EP-0293978-A2 (1H-azol-1-ylmethyl)substituted benzotriazole derivatives JANSSEN PHARMACEUTICA N.V. (BE) 1988-12-07 EP disclosed