SCHEMBL9524501

SCHEMBL9524501

COC(=O)CC[C@@H](NC(=O)c1ccc(Br)cc1Cl)C(=O)OC

nearest known ligand 0.46

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.46
MAPK1 P28482 1/20 0.46
ITGB1 P05556 1/20 0.44
ITGA4 P13612 1/20 0.44
TAS1R3 Q7RTX0 2/20 0.44
TAS1R1 Q7RTX1 2/20 0.44
ALOX5 P09917 1/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
HPGD P15428 4/20 0.41
CLPP Q16740 2/20 0.41
FLT1 P17948 1/20 0.40
FLT4 P35916 1/20 0.40
KDR P35968 1/20 0.40
HDAC1 Q13547 2/20 0.40
HDAC6 Q9UBN7 2/20 0.40
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524496 1.00 ALDH1A1 (0.46) ALDH1A1MAPK1ITGB1ITGA4TAS1R3
SCHEMBL13923473 0.84 ITGB1 (0.47) ALDH1A1MAPK1ITGB1ITGA4TAS1R3
SCHEMBL16898779 0.83 ALDH1A1 (0.44) ALDH1A1MAPK1TAS1R3TAS1R1ALOX5
SCHEMBL18241389 0.83 ALDH1A1 (0.44) ALDH1A1MAPK1TAS1R3TAS1R1ALOX5
SCHEMBL16898289 0.80 L3MBTL1 (0.55) TAS1R3TAS1R1ALOX5CA12CA1
SCHEMBL16898288 0.80 L3MBTL1 (0.55) TAS1R3TAS1R1ALOX5CA12CA1
SCHEMBL8819401 0.80 CA12 (0.43) ALDH1A1MAPK1TAS1R3TAS1R1ALOX5
SCHEMBL8819411 0.80 CA12 (0.43) ALDH1A1MAPK1TAS1R3TAS1R1ALOX5
SCHEMBL10654280 0.78 ALDH1A1 (0.49) ALDH1A1HPGDFLT1FLT4KDR
SCHEMBL10570037 0.78 ITGB1 (0.55) ITGB1ITGA4CA1CA2HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0327190-B1 Pyrido(2,3-d)pyrimidine derivatives UNIV PRINCETON (US) 1993-12-08 EP disclosed
EP-0327190-A1 Pyrido(2,3-d)pyrimidine derivatives THE TRUSTEES OF PRINCETON UNIVERSITY (US) 1989-08-09 EP disclosed