SCHEMBL9524767

SCHEMBL9524767

CCCCN(CCOc1cccc2ccccc12)C(=O)OCCNC(=O)c1cncc(Br)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.53
NPC1 O15118 3/20 0.49
RAB9A P51151 3/20 0.49
ALDH1A1 P00352 4/20 0.48
SMN1; SMN2 Q16637 3/20 0.48
POLB P06746 1/20 0.46
NPSR1 Q6W5P4 1/20 0.45
HTR1B P28222 2/20 0.45
CYP1A2 P05177 2/20 0.44
CYP3A4 P08684 2/20 0.44
CYP2C19 P33261 2/20 0.44
CYP2C9 P11712 1/20 0.44
HTT P42858 1/20 0.44
HTR1D P28221 1/20 0.43
KDM4E B2RXH2 1/20 0.42
HPGD P15428 1/20 0.42
GLA P06280 1/20 0.41
MAPT P10636 1/20 0.41
PKM P14618 1/20 0.39
MEN1 O00255 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525271 0.89 NPC1 (0.52) LMNANPC1RAB9AALDH1A1SMN1; SMN2
Iodide SCHEMBL9526181 0.85 HTR1B (0.43) LMNANPC1ALDH1A1HTR1BCYP2C9
Iodide SCHEMBL9525064 0.84 HTR1B (0.42) LMNANPC1ALDH1A1HTR1BCYP2C9
SCHEMBL9528248 0.82 LMNA (0.62) LMNANPC1RAB9AALDH1A1SMN1; SMN2
SCHEMBL9526235 0.82 LMNA (0.49) LMNANPC1RAB9AALDH1A1SMN1; SMN2
Iodide SCHEMBL9525497 0.77 HPGD (0.41) LMNANPC1RAB9AALDH1A1SMN1; SMN2
Iodide SCHEMBL9526359 0.75 HTR1B (0.40) LMNANPC1ALDH1A1HTR1BHTR1D
Iodide SCHEMBL9525321 0.75 HTR1B (0.41) LMNANPC1RAB9AALDH1A1HTR1B
Iodide SCHEMBL9528189 0.74 HPGD (0.42) LMNANPC1ALDH1A1HTR1BHTR1D
Iodide SCHEMBL9525155 0.73 HPGD (0.44) LMNANPC1ALDH1A1HTR1BHTR1D

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed