SCHEMBL9524912

SCHEMBL9524912

CCOC(=O)C(=Cc1ccccc1Cl)C(=O)c1ccc(-n2c(C)nc3cnccc32)cc1

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
POLB P06746 2/20 0.39
ALDH1A1 P00352 1/20 0.39
HSD17B10 Q99714 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525015 0.92 TP53 (0.40) MEN1KMT2AHSD17B10
SCHEMBL9525496 0.78 MAPT (0.53) MEN1KMT2AALDH1A1HSD17B10
SCHEMBL9726988 0.77 KMT2A (0.43) MEN1KMT2APOLBALDH1A1
SCHEMBL9524574 0.75 MAPT (0.47) MEN1KMT2APOLBALDH1A1HSD17B10
SCHEMBL9727194 0.73 TP53 (0.46) MEN1KMT2AALDH1A1HSD17B10
SCHEMBL7869540 0.72 MEN1 (0.46) MEN1KMT2AHSD17B10
SCHEMBL9868470 0.72 TP53 (0.40)
SCHEMBL9524966 0.72 TP53 (0.46) MEN1KMT2AHSD17B10
SCHEMBL9524668 0.71 HSD17B10 (0.55) MEN1KMT2AHSD17B10
SCHEMBL9524861 0.71 TP53 (0.39) MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0466711-B1 DIHYDROPYRIMIDINE ANTIALLERGY AGENTS PFIZER LTD (GB) 1993-10-27 EP disclosed
EP-0462986-B1 IMIDAZOPYRIMIDINE ANTIALLERGY AGENTS Pfizer Limited (GB) 1993-10-06 EP disclosed
US-5250531-A Antiallergens, antiinflammatory agents PFIZER INC. (US) 1993-10-05 US disclosed
EP-0530207-A1 IMIDAZOPYRIDINE PAF ANTAGONISTS Pfizer Limited (GB) 1993-03-10 EP disclosed
EP-0466711-A1 DIHYDROPYRIMIDINE ANTIALLERGY AGENTS. PFIZER LTD (GB) 1992-01-22 EP disclosed
EP-0462986-A1 IMIDAZOPYRIMIDINE ANTIALLERGY AGENTS. PFIZER LTD (GB) 1992-01-02 EP disclosed
WO-1991017162-A1 IMIDAZOPYRIDINE PAF ANTAGONISTS PFIZER LIMITED (GB) 1991-11-14 WO disclosed
WO-1990011281-A1 DIHYDROPYRIMIDINE ANTIALLERGY AGENTS PFIZER LIMITED (GB) 1990-10-04 WO disclosed
WO-1990010632-A1 IMIDAZOPYRIMIDINE ANTIALLERGY AGENTS PFIZER LIMITED (GB) 1990-09-20 WO disclosed