SCHEMBL9524934

SCHEMBL9524934

COC(=O)c1cc2ccc3ccccc3c2s1

nearest known ligand 0.66

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 6/20 0.66
HPGD P15428 6/20 0.66
KDM4E B2RXH2 8/20 0.61
MAPT P10636 5/20 0.61
RAB9A P51151 3/20 0.61
NPC1 O15118 2/20 0.61
NPSR1 Q6W5P4 2/20 0.61
L3MBTL1 Q9Y468 3/20 0.61
ATM Q13315 3/20 0.61
CASP3 P42574 1/20 0.61
SMN1; SMN2 Q16637 1/20 0.61
SENP7 Q9BQF6 1/20 0.61
SENP6 Q9GZR1 1/20 0.61
TDP1 Q9NUW8 1/20 0.61
MEN1 O00255 2/20 0.45
KMT2A Q03164 2/20 0.45
NCEH1 Q6PIU2 1/20 0.43
HSD17B10 Q99714 3/20 0.42
POLB P06746 1/20 0.42
MAPK1 P28482 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30020347 0.84 KDM4E (0.83) ALDH1A1HPGDKDM4EMAPTRAB9A
SCHEMBL7461107 0.83 KDM4E (0.68) ALDH1A1HPGDKDM4EMAPTRAB9A
SCHEMBL11561435 0.82 MAPT (0.61) ALDH1A1HPGDKDM4EMAPTRAB9A
SCHEMBL9431295 0.80 ALDH1A1 (0.60) ALDH1A1HPGDKDM4EMAPTRAB9A
SCHEMBL15384380 0.79 HPGD (0.55) ALDH1A1HPGDKDM4EMAPTRAB9A
SCHEMBL2895989 0.79 ALDH1A1 (0.55) ALDH1A1HPGDKDM4EMAPTL3MBTL1
SCHEMBL5125588 0.79 HPGD (0.55) ALDH1A1HPGDKDM4EMAPTRAB9A
SCHEMBL28540745 0.79 KDM4E (0.61) ALDH1A1HPGDKDM4EMAPTRAB9A
SCHEMBL9526183 0.79 HPGD (0.55) ALDH1A1HPGDKDM4EMAPTRAB9A
SCHEMBL25094033 0.78 HDAC1 (0.56) ALDH1A1HPGDKDM4EMAPTRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0183439-B1 POLYCYCLIC COMPOUNDS, THEIR PREPARATION AND USE AND FORMULATIONS CONTAINING THEM THE WELLCOME FOUNDATION LIMITED (GB) 1993-02-03 EP disclosed
US-5075455-A Microbiocides, antitumor agents BURROUGHS WELLCOME CO. (US) 1991-12-24 US disclosed
US-5049581-A Dibenzofurans having anti-tumor activity BURROUGHS WELLCOME CO. (US) 1991-09-17 US disclosed
US-5017600-A Antitumor BURROUGHS WELLCOME CO. (US) 1991-05-21 US disclosed
US-5008286-A Antitumor agents BURROUGHS WELLCOME CO. (US) 1991-04-16 US disclosed
US-4970227-A ANTITUMOR BURROUGHS WELLCOME CO. (US) 1990-11-13 US disclosed
US-4965285-A ANTITUMOR AGENTS BURROUGHS WELLCOME CO. (US) 1990-10-23 US disclosed
US-4866070-A ANTITUMOR AGENT BURROUGHS WELLCOME CO. (US) 1989-09-12 US disclosed
EP-0183439-A2 Polycyclic compounds, their preparation and use and formulations containing them THE WELLCOME FOUNDATION LIMITED (GB) 1986-06-04 EP disclosed