SCHEMBL28540745

SCHEMBL28540745

NC(=O)c1cc2ccc3ccccc3c2s1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.61
RAB9A P51151 3/20 0.61
MAPT P10636 3/20 0.61
NPC1 O15118 2/20 0.61
NPSR1 Q6W5P4 1/20 0.61
TDP1 Q9NUW8 2/20 0.51
L3MBTL1 Q9Y468 2/20 0.51
CASP3 P42574 1/20 0.51
ATM Q13315 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.51
SENP7 Q9BQF6 1/20 0.51
SENP6 Q9GZR1 1/20 0.51
CNR1 P21554 1/20 0.43
CNR2 P34972 1/20 0.43
MAP2K1 Q02750 2/20 0.41
CHEK1 O14757 2/20 0.41
AURKA O14965 2/20 0.41
DAPK3 O43293 2/20 0.41
PIM1 P11309 2/20 0.41
FGFR1 P11362 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7461107 0.84 KDM4E (0.68) KDM4ERAB9AMAPTNPC1NPSR1
Hydrochloric Acid SCHEMBL9431489 0.83 KDM4E (0.54) KDM4ERAB9AMAPTNPC1NPSR1
SCHEMBL11561435 0.83 MAPT (0.61) KDM4ERAB9AMAPTNPC1NPSR1
SCHEMBL9524934 0.79 ALDH1A1 (0.66) KDM4ERAB9AMAPTNPC1NPSR1
SCHEMBL28537323 0.78 LIMK1 (0.48) KDM4EMAPTTDP1L3MBTL1CNR1
SCHEMBL13295842 0.76 CHRNA1 (0.48) KDM4ERAB9AMAPTNPC1NPSR1
SCHEMBL30020347 0.75 KDM4E (0.83) KDM4ERAB9AMAPTNPC1NPSR1
SCHEMBL347544 0.74 BCL2L1 (0.69) RAB9AL3MBTL1CASP3SENP7SENP6
SCHEMBL29366392 0.74 BCL2L1 (0.69) RAB9AL3MBTL1CASP3SENP7SENP6
Hydrochloric Acid SCHEMBL2196804 0.73 BCL2L1 (0.67) RAB9AL3MBTL1CASP3SENP7SENP6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108727416-B Tricyclic heteroaromatic amide derivative and preparation and application thereof 北京大学 2021-03-09 CN disclosed