SCHEMBL9525217

SCHEMBL9525217

COc1cccc(N(CCO)C(=O)c2cncc(Br)c2)c1

nearest known ligand 0.50

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 1/20 0.47
DGAT2 Q96PD7 1/20 0.43
ALDH1A1 P00352 2/20 0.43
HPGD P15428 1/20 0.43
OPRM1 P35372 1/20 0.43
OPRD1 P41143 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.42
MTNR1A P48039 4/20 0.42
MTNR1B P49286 4/20 0.42
HSD17B2 P37059 2/20 0.41
HSD17B1 P14061 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
ROCK2 O75116 2/20 0.41
LIMK1 P53667 1/20 0.41
ROCK1 Q13464 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9525689 0.81 KMT2A (0.51) KMT2AALDH1A1OPRM1OPRD1SMN1; SMN2
SCHEMBL9524476 0.80 HTT (0.45) KMT2AALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL9524632 0.79 HTT (0.47) KMT2AALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL9525452 0.78 HTT (0.56) KMT2ASMN1; SMN2NPC1RAB9A
SCHEMBL9524303 0.77 HTT (0.50) KMT2AALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL9525869 0.76 HTT (0.44) KMT2AALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL9525530 0.76 HTT (0.46) KMT2AALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL9526168 0.76 HTT (0.46) KMT2AALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL9525423 0.76 EGFR (0.47) KMT2AALDH1A1SMN1; SMN2NPC1RAB9A
SCHEMBL9524339 0.76 EGFR (0.47) KMT2AALDH1A1SMN1; SMN2NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0301751-B1 PYRIDINIUM DERIVATIVES, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 1993-03-10 EP disclosed
US-4962113-A PLATELET ACTIVATING FACTOR ANTAGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD (JP) 1990-10-09 US disclosed
EP-0301751-A1 Pyridinium derivatives, their production and use Takeda Chemical Industries, Ltd. (JP) 1989-02-01 EP disclosed