SCHEMBL9525659

SCHEMBL9525659

CC1(C)CC(c2ccc(-c3ccccc3)cn2)c2cc(C#N)ccc2O1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 8/20 0.44
ABCB1 P08183 7/20 0.39
CTSD P07339 1/20 0.36
BACE1 P56817 1/20 0.36
GABRA1 P14867 1/20 0.36
GABRG2 P18507 1/20 0.36
GABRB3 P28472 1/20 0.36
GABRA5 P31644 1/20 0.36
GABRA3 P34903 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9524618 0.85 ABCB1 (0.41) ABCC9ABCB1
SCHEMBL9524383 0.84 ABCC9 (0.43) ABCC9ABCB1
SCHEMBL9525156 0.84 ABCB1 (0.38) ABCC9ABCB1
SCHEMBL8338287 0.84 ABCC9 (0.43) ABCC9ABCB1
SCHEMBL8967989 0.84 ABCC9 (0.43) ABCC9ABCB1
SCHEMBL9524429 0.82 ABCC9 (0.44) ABCC9ABCB1
SCHEMBL9525734 0.81 KDM4E (0.37) ABCC9ABCB1
SCHEMBL9524678 0.79 ABCC9 (0.45) ABCC9ABCB1
SCHEMBL9523930 0.79 ABCC9 (0.40) ABCC9ABCB1
SCHEMBL9524801 0.78 ABCC9 (0.45) ABCC9ABCB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0298452-B1 2H-1-BENZOPYRANE DERIVATIVES SUBSTITUTED IN POSITION 4 BY ARYL OR N-HETEROARYL F. HOFFMANN-LA ROCHE AG (CH) 1993-06-30 EP disclosed
US-5118694-A Hypotensive agents; treatment for cardiovascular and muscular disorders HOFFMANN-LA ROCHE INC. (US) 1992-06-02 US disclosed
US-4971982-A HYPOTENSIVE AGENTS, CARDIOVASCULAR DISORDERS, SMOOTH MUSCLE DISORDERS HOFFMANN-LA ROCHE INC. (US) 1990-11-20 US disclosed
EP-0298452-A2 2H-1-benzopyrane derivatives substituted in position 4 by aryl or N-heteroaryl F. HOFFMANN-LA ROCHE AG (CH) 1989-01-11 EP disclosed