SCHEMBL9526082

SCHEMBL9526082

COc1ccnc(CSc2nc3cc(OC)c(OC(F)(F)F)cc3[nH]2)c1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
NOS2 P35228 4/20 0.62
NOS3 P29474 3/20 0.62
NOS1 P29475 3/20 0.62
CYP2E1 P05181 15/20 0.53
CYP2C8 P10632 15/20 0.53
CYP2D6 P10635 15/20 0.53
CYP2C9 P11712 15/20 0.53
CYP2B6 P20813 15/20 0.53
CYP2C19 P33261 15/20 0.53
CYP3A4 P08684 14/20 0.53
CYP1A2 P05177 13/20 0.53
BRS3 P32247 1/20 0.45
ENPP1 P22413 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9528059 0.98 NOS2 (0.65) NOS2NOS3NOS1CYP2E1CYP2C8
SCHEMBL9527996 0.91 NOS2 (0.59) NOS2NOS3NOS1CYP2E1CYP2C8
SCHEMBL9527723 0.89 NOS2 (0.61) NOS2NOS3NOS1CYP2E1CYP2C8
SCHEMBL9686697 0.89 NOS2 (0.56) NOS2NOS3NOS1CYP2E1CYP2C8
SCHEMBL9526158 0.86 NOS2 (0.62) NOS2NOS3NOS1CYP2E1CYP2C8
SCHEMBL9527785 0.86 NOS2 (0.68) NOS2NOS3NOS1CYP2E1CYP2C8
SCHEMBL9526760 0.84 NOS2 (0.65) NOS2NOS3NOS1CYP2E1CYP2C8
SCHEMBL9528045 0.83 ENPP1 (0.44) NOS2NOS3NOS1CYP2E1CYP2C8
SCHEMBL9528042 0.82 CYP1A2 (0.56) NOS2NOS3NOS1CYP2E1CYP2C8
SCHEMBL9526119 0.82 CYP2E1 (0.46) NOS2NOS3NOS1CYP2E1CYP2C8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0134400-B1 FLUOROALKOXYSUBSTITUTED PYRIDYLMETHYLTHIO-(OR SULFINYL-)BENZIMIDAZOLES HAVING A SECRETOLYTIC ACTIVITY Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1993-03-24 EP disclosed
US-4555518-A ANTIULCER AGENTS BYK GULDEN LOMBERG CHEMISCHE FABRIK GMBH (DE) 1985-11-26 US disclosed
EP-0134400-A2 Fluoroalkoxysubstituted pyridylmethylthio-(or sulfinyl-)benzimidazoles having a secretolytic activity Byk Gulden Lomberg Chemische Fabrik GmbH (DE) 1985-03-20 EP disclosed