SCHEMBL9526213

SCHEMBL9526213

O=C(CCl)c1cc(Cl)ccc1Cl

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.71
MAPK1 P28482 1/20 0.71
HIF1A Q16665 1/20 0.71
ERCC5 P28715 2/20 0.62
FEN1 P39748 2/20 0.62
TP53 P04637 2/20 0.61
LMNA P02545 3/20 0.53
MAPT P10636 1/20 0.53
GSK3B P49841 3/20 0.52
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
HPGD P15428 1/20 0.49
CYP2C19 P33261 1/20 0.49
SMN1; SMN2 Q16637 2/20 0.47
GAA P10253 1/20 0.47
NFKB1 P19838 1/20 0.47
NFKB2 Q00653 1/20 0.47
RELA Q04206 1/20 0.47
TSHR P16473 2/20 0.45
CASP1 P29466 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1427082 0.84 ERCC5 (0.59) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL4449153 0.83 ERCC5 (0.62) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL29481555 0.83 ALDH1A1 (1.00) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL1691536 0.83 ALDH1A1 (1.00) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL404490 0.82 ERCC5 (0.61) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL29391618 0.82 ERCC5 (0.61) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL1154685 0.82 MAPK1 (0.63) ALDH1A1MAPK1HIF1ATP53LMNA
SCHEMBL11613851 0.82 ALDH1A1 (0.61) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL21055979 0.82 ALDH1A1 (0.53) ALDH1A1MAPK1HIF1AERCC5FEN1
SCHEMBL16770754 0.82 ERCC5 (0.61) ALDH1A1MAPK1HIF1AERCC5FEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101243081-A Pyrido[2,3-d]pyrimidine-2,4-diamine compounds as PTP1B inhibitors HOFFMANN LA ROCHE (CH) 2008-08-13 CN disclosed
EP-0365913-B1 Substituted 2-aminothiazoles BAYER AG (DE) 1993-11-18 EP disclosed
US-5104879-A ANTIMYCOTICALLY ACTIVE SUBSTITUTED 2-AMINOTHIAZOLES BAYER AKTIENGESELLSCHAFT (DE) 1992-04-14 US disclosed
EP-0365913-A2 Substituted 2-aminothiazoles BAYER AG (DE) 1990-05-02 EP disclosed